SCHEMBL6498709

SCHEMBL6498709

Cc1sc(-c2ccc(F)c(Cl)c2)nc1C(=O)NCc1cc(CC(OC(C)C)C(=O)OC(=O)C(F)(F)F)ccn1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 5/20 0.34
GSK3B P49841 5/20 0.34
KMO O15229 1/20 0.33
NPC1 O15118 1/20 0.33
WDR5 P61964 2/20 0.32
MAPK1 P28482 2/20 0.32
PPARA Q07869 2/20 0.32
PPARD Q03181 1/20 0.32
ROS1 P08922 1/20 0.31
ALK Q9UM73 1/20 0.31
SUCNR1 Q9BXA5 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
RHOC P08134 1/20 0.31
RHOA P61586 1/20 0.31
P2RX7 Q99572 1/20 0.31
KLKB1 P03952 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6504395 0.93 PPARA (0.37) CDK2GSK3BWDR5PPARAPPARD
SCHEMBL6505045 0.90 SMN1; SMN2 (0.35) NPC1PPARAPPARDTP53
Trifluoroacetic Acid SCHEMBL6498705 0.90 PPARA (0.37) CDK2GSK3BPPARAPPARD
SCHEMBL6531507 0.89 PARP1 (0.36) NPC1MAPK1PPARAPPARDMAPT
SCHEMBL6494741 0.88 PPARA (0.39) CDK2GSK3BWDR5PPARAPPARD
SCHEMBL6495822 0.88 SHMT1 (0.39) WDR5MAPTKLKB1
SCHEMBL6505593 0.87 ADORA2A (0.35) NPC1PPARAPPARD
SCHEMBL6503597 0.83 KDM4E (0.36) NPC1MAPTKLKB1
Trifluoroacetic Acid SCHEMBL6504387 0.83 PPARA (0.42) PPARAPPARDRHOCRHOA
SCHEMBL6499174 0.82 ADORA1 (0.38) NPC1WDR5MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed