SCHEMBL6505045

SCHEMBL6505045

Cc1ccc(-c2nc(C(=O)NCc3cc(CC(OC(C)C)C(=O)OC(=O)C(F)(F)F)ccn3)c(C)s2)cc1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
PPARA Q07869 9/20 0.34
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
PPARD Q03181 4/20 0.33
PPARG P37231 3/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
ROCK2 O75116 1/20 0.32
KMT2A Q03164 1/20 0.32
HTT P42858 1/20 0.32
IKBKE Q14164 1/20 0.32
TBK1 Q9UHD2 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6504395 0.94 PPARA (0.37) SMN1; SMN2PPARAPPARDPPARG
SCHEMBL6531507 0.94 PARP1 (0.36) SMN1; SMN2NPC1RAB9APPARAADORA2A
SCHEMBL6494741 0.93 PPARA (0.39) PPARAADORA2AADORA1PPARDPPARG
SCHEMBL6498709 0.90 CDK2 (0.34) NPC1PPARAPPARDTP53
Trifluoroacetic Acid SCHEMBL6505042 0.89 PPARA (0.42) SMN1; SMN2NPC1RAB9APPARAPPARD
SCHEMBL6503597 0.88 KDM4E (0.36) NPC1RAB9AKDM4EALDH1A1KMT2A
SCHEMBL6505593 0.87 ADORA2A (0.35) NPC1RAB9APPARAADORA2AADORA1
SCHEMBL6495822 0.86 SHMT1 (0.39) KDM4EHPGDKMT2A
SCHEMBL6499174 0.86 ADORA1 (0.38) SMN1; SMN2NPC1RAB9AADORA2AADORA1
Trifluoroacetic Acid SCHEMBL6531504 0.83 PPARA (0.40) SMN1; SMN2PPARAPPARDPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed