SCHEMBL6551937

SCHEMBL6551937

CC(C)Oc1nn(-c2ccc(S(=O)(=O)NC3CC(C)(C)NC(C)(C)C3)cc2)c(=O)o1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.50
MEN1 O00255 1/20 0.50
MAPT P10636 1/20 0.47
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ABHD16A O95870 1/20 0.37
POLB P06746 2/20 0.36
RAB9A P51151 1/20 0.36
IKBKB O14920 1/20 0.36
LPL P06858 1/20 0.35
LIPC P11150 1/20 0.35
LIPE Q05469 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6551927 0.90 KMT2A (0.52) KMT2AMEN1MAPTALDH1A1TSHR
SCHEMBL6551189 0.84 ALDH1A1 (0.41) KMT2AMEN1ALDH1A1ABHD16ALPL
SCHEMBL6551212 0.74 ABHD16A (0.41) KMT2AABHD16ALPLLIPCLIPE
SCHEMBL6552668 0.74 ABHD16A (0.46) KMT2AMEN1ALDH1A1TSHRABHD16A
SCHEMBL27996013 0.69 KMT2A (0.76) KMT2AMEN1MAPTALDH1A1TSHR
SCHEMBL23052367 0.66 KMT2A (1.00) KMT2AMEN1MAPTALDH1A1TSHR
SCHEMBL23045690 0.66 KMT2A (0.70) KMT2AMEN1MAPTALDH1A1TSHR
SCHEMBL6551932 0.65 ABHD16A (0.53) ABHD16ALPLLIPCLIPE
SCHEMBL7044899 0.64 MGLL (0.59) ABHD16ALPLLIPCLIPE
SCHEMBL7046480 0.64 ABHD16A (0.50) MAPTALDH1A1ABHD16APOLBLPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1482929-A1 USE OF SUBSTITUTED 3-PHENYL-5-ALKOXY-1,3,4-OXDIAZOLE-2-ONE FOR PRODUCING MEDICAMENTS THAT INHIBIT PANCREATIC LIPASE Aventis Pharma Deutschland GmbH (DE) 2004-12-08 EP disclosed
US-20030236288-A1 Use of substituted 3-phenyl-5-alkoxy-3H-(1,3,4)-oxadizol-2-ones for inhibiting pancreatic lipase AVENTIS PHARMA DEUTSCHLAND GMBH 2003-12-25 US disclosed
EP-1214302-B1 SUBSTITUTED 3-PHENYL-5-ALKOXI-1,3,4-OXDIAZOL-2-ONES AND THEIR USE AS LIPASE INHIBITORS AVENTIS PHARMA GMBH (DE) 2003-10-29 EP disclosed
WO-2003072098-A1 USE OF SUBSTITUTED 3-PHENYL-5-ALKOXY-1,3,4-OXDIAZOLE-2-ONE FOR PRODUCING MEDICAMENTS THAT INHIBIT PANCREATIC LIPASE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-09-04 WO disclosed
US-6596742-B1 Inhibitory effect on the hormone-sensitive lipase, HSL. insecticides, controlling metabolism and multistage synthesis AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-07-22 US disclosed
EP-1214302-A1 SUBSTITUTED 3-PHENYL-5-ALKOXI-1,3,4-OXDIAZOL-2-ONES AND THEIR USE AS LIPASE INHIBITORS Aventis Pharma Deutschland GmbH (DE) 2002-06-19 EP disclosed
WO-2001017981-A1 SUBSTITUTED 3-PHENYL-5-ALKOXI-1,3,4-OXDIAZOL-2-ONES AND THEIR USE AS LIPASE INHIBITORS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-03-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030236288-A1 Use of substituted 3-phenyl-5-alkoxy-3H-(1,3,4)-oxadizol-2-ones for inhibiting pancreatic lipase PNLIP, CEL, LIPE KMT2A 3097/4885MEN1 4309/4885MAPT 4762/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.