SCHEMBL6561734

SCHEMBL6561734

CN(C)C(=O)c1csc(CC(=O)O)c1Cl

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
HPGD P15428 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HTT P42858 1/20 0.33
PTGDR2 Q9Y5Y4 2/20 0.33
GSK3B P49841 1/20 0.33
MAPT P10636 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
GABRA5 P31644 1/20 0.30
GABRB2 P47870 1/20 0.30
HSD17B10 Q99714 1/20 0.30
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2655191 0.74 PTGDR2 (0.40) ALDH1A1MEN1KMT2APTGDR2KEAP1
SCHEMBL7042949 0.70 ALDH1A1 (0.32) ALDH1A1MEN1KMT2AHPGDSMN1; SMN2
SCHEMBL28007558 0.68 THRB (0.34) ALDH1A1MEN1KMT2APTGDR2MAPT
SCHEMBL7904931 0.67 ALDH1A1 (0.35) ALDH1A1MEN1KMT2AHPGDSMN1; SMN2
SCHEMBL22615007 0.65 ALDH1A1 (0.57) ALDH1A1MEN1KMT2AHPGDHTT
SCHEMBL27565970 0.63 GABRA5 (0.42) ALDH1A1MEN1KMT2AHPGDPTGDR2
SCHEMBL5797600 0.62 CA2 (0.33)
SCHEMBL827254 0.62 GSK3B (0.52) ALDH1A1MEN1KMT2AHPGDSMN1; SMN2
SCHEMBL18301798 0.62 BCAT2 (0.57) MEN1KMT2ASMN1; SMN2KEAP1AKR1B1
SCHEMBL19178089 0.62 KEAP1 (0.42) MEN1KMT2AMAPTKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904079-B1 ANTIDIABETIC AGENTS MERCK & CO INC (US) 2004-03-24 EP disclosed
EP-0904079-A4 1999-05-06 EP disclosed
EP-0904079-A1 ANTIDIABETIC AGENTS Merck & Co., Inc. (US) 1999-03-31 EP disclosed
US-5859051-A ACETYLPHENOL DERIVATIVES MERCK & CO., INC. (US) 1999-01-12 US disclosed
WO-1997027857-A1 ANTIDIABETIC AGENTS MERCK & CO., INC. (US) 1997-08-07 WO disclosed