SCHEMBL6561813

SCHEMBL6561813

CN(C)CCN(C)C(=O)c1ccc(C#CCNc2ccc(C(=N)NC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.42
ACACB O00763 3/20 0.35
PTGES O14684 1/20 0.33
HDAC4 P56524 1/20 0.32
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
PIK3CA P42336 3/20 0.32
MTOR P42345 3/20 0.32
PIK3CG P48736 3/20 0.32
ATR Q13535 1/20 0.32
MCHR1 Q99705 1/20 0.32
DRD2 P14416 1/20 0.31
NR3C2 P08235 1/20 0.31
KCNH2 Q12809 1/20 0.31
NAMPT P43490 2/20 0.31
ROCK2 O75116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563283 0.89 PTPN11 (0.46) PTPN11ACACBPTGESATR
SCHEMBL6563495 0.84 PTPN11 (0.36) PTPN11ACACBPTGESCCNCCDK8
SCHEMBL6563749 0.81 ITGB3 (0.41) ACACBATR
SCHEMBL6563355 0.80 PTPN11 (0.47) PTPN11PTGES
SCHEMBL6563070 0.80 PTPN11 (0.44) PTPN11NAMPT
SCHEMBL6563526 0.79 PTPN11 (0.38) PTPN11ACACBPTGES
SCHEMBL6561879 0.79 PTPN11 (0.38) PTPN11ACACBPTGES
SCHEMBL7674981 0.78 ABL1 (0.43) PTPN11ACACBNAMPT
SCHEMBL7686729 0.78 PTPN11 (0.43) PTPN11ACACBNAMPT
SCHEMBL6561858 0.77 GRM5 (0.47) PTPN11NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed