SCHEMBL6561858

SCHEMBL6561858

CC1CCN(C(=O)c2ccc(C#CCNc3ccc(C(=N)NC(=O)OC(C)(C)C)cc3)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.47
HPGD P15428 3/20 0.41
NAMPT P43490 1/20 0.41
ABL1 P00519 1/20 0.41
RIN1 Q13671 1/20 0.41
PTPN11 Q06124 1/20 0.40
HRH3 Q9Y5N1 4/20 0.40
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
GRM3 Q14832 1/20 0.39
ACHE P22303 1/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674981 0.91 ABL1 (0.43) HPGDNAMPTABL1RIN1PTPN11
SCHEMBL7686729 0.91 PTPN11 (0.43) GRM5HPGDNAMPTABL1RIN1
SCHEMBL6565384 0.89 GRM5 (0.46) GRM5HPGDNAMPTABL1RIN1
SCHEMBL6563002 0.86 HRH3 (0.42) GRM5HPGDNAMPTPTPN11HRH3
SCHEMBL6563511 0.83 PTPN11 (0.40) PTPN11GRM3POLBHSD11B1
SCHEMBL6563920 0.82 KLK5 (0.41) PTPN11KMT2AALDH1A1
SCHEMBL6565248 0.82 GRM5 (0.56) GRM5HPGDHRH3CRHBPCRHR2
SCHEMBL6565533 0.81 ACACB (0.45) ABL1RIN1PTPN11KMT2AALDH1A1
SCHEMBL6561810 0.80 HSD11B1 (0.40) ABL1RIN1PTPN11ACHEALDH1A1
SCHEMBL6565229 0.79 PTPN11 (0.34) PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed