SCHEMBL6563511

SCHEMBL6563511

CC(C)(C)OC(=O)NC(=N)c1ccc(NCC#Cc2ccc(C(=O)N3CCCC3CO)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.40
SPHK2 Q9NRA0 3/20 0.38
POLB P06746 2/20 0.37
ROCK2 O75116 1/20 0.36
NPC1 O15118 1/20 0.35
SPHK1 Q9NYA1 3/20 0.35
GRM3 Q14832 3/20 0.35
PDK2 Q15119 1/20 0.35
USP1 O94782 1/20 0.34
HSD11B1 P28845 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563002 0.90 HRH3 (0.42) PTPN11NPC1HSD11B1
SCHEMBL6563920 0.88 KLK5 (0.41) PTPN11ROCK2NPC1PDK2
SCHEMBL7674981 0.84 ABL1 (0.43) PTPN11POLB
SCHEMBL7686729 0.84 PTPN11 (0.43) PTPN11
SCHEMBL6565962 0.83 SPHK2 (0.41) SPHK2POLBROCK2SPHK1GRM3
SCHEMBL6561858 0.83 GRM5 (0.47) PTPN11POLBGRM3HSD11B1
SCHEMBL6563779 0.82 KCNK3 (0.38) PTPN11HSD11B1
SCHEMBL6565417 0.81 PTPN11 (0.36) PTPN11NPC1HSD11B1
SCHEMBL6565384 0.81 GRM5 (0.46) PTPN11POLBNPC1
SCHEMBL6561835 0.80 PTPN11 (0.35) PTPN11NPC1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed