SCHEMBL6563920

SCHEMBL6563920

COC(=O)C1CCCN1C(=O)c1ccc(C#CCNc2ccc(C(=N)NC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.41
PTPN11 Q06124 1/20 0.39
NPC1 O15118 2/20 0.39
ROCK2 O75116 1/20 0.39
PDK2 Q15119 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MMP2 P08253 2/20 0.37
MMP9 P14780 2/20 0.37
MMP8 P22894 2/20 0.37
MMP13 P45452 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
LOX P28300 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563002 0.89 HRH3 (0.42) PTPN11NPC1ALDH1A1
SCHEMBL6563511 0.88 PTPN11 (0.40) PTPN11NPC1ROCK2PDK2
SCHEMBL6563770 0.84 SPHK1 (0.43) NPC1PDK2ALDH1A1MMP2MMP9
SCHEMBL7686729 0.83 PTPN11 (0.43) PTPN11ALDH1A1KMT2AL3MBTL1
SCHEMBL7674981 0.83 ABL1 (0.43) PTPN11ALDH1A1KMT2AL3MBTL1
SCHEMBL6561858 0.82 GRM5 (0.47) PTPN11ALDH1A1KMT2A
SCHEMBL6565417 0.81 PTPN11 (0.36) PTPN11NPC1ALDH1A1
SCHEMBL6565384 0.80 GRM5 (0.46) PTPN11NPC1KMT2A
SCHEMBL6561835 0.78 PTPN11 (0.35) PTPN11NPC1ALDH1A1KMT2A
SCHEMBL6563591 0.78 LRRK2 (0.39) ROCK2PDK2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed