SCHEMBL6563299

SCHEMBL6563299

Cc1cc(C#CCNc2ccc(C(=N)NC(=O)OC(C)(C)C)cc2)ccc1C(=O)N1CCC(NC(=O)OC(C)(C)C)C1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.40
PARP1 P09874 1/20 0.39
ADORA2A P29274 3/20 0.38
ADORA3 P0DMS8 2/20 0.38
ADORA2B P29275 2/20 0.38
CFTR P13569 1/20 0.38
HSD11B1 P28845 5/20 0.37
CYP2C9 P11712 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
BRD4 O60885 1/20 0.36
KDM4D Q6B0I6 2/20 0.35
CTSK P43235 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
MCL1 Q07820 1/20 0.35
ACACB O00763 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565379 0.90 USP30 (0.43) PARP1HSD11B1CYP2C9
SCHEMBL6565533 0.87 ACACB (0.45) HSD11B1ACACB
SCHEMBL6561973 0.85 JAK1 (0.38) ACACB
SCHEMBL6565417 0.84 PTPN11 (0.36) NAMPTHSD11B1ACACB
SCHEMBL6565215 0.81 PIK3CA (0.38) ACACB
SCHEMBL6561810 0.80 HSD11B1 (0.40) HSD11B1ACACB
SCHEMBL6565339 0.80 HPGD (0.39) HSD11B1CYP2C9ACACB
SCHEMBL6563779 0.79 KCNK3 (0.38) HSD11B1
SCHEMBL6563395 0.79 PTPN11 (0.35)
SCHEMBL6561858 0.79 GRM5 (0.47) NAMPTHSD11B1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed