SCHEMBL6565441

SCHEMBL6565441

N#Cc1ccc(NCC#Cc2ccc(C(=O)c3ccccn3)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
GRM4 Q14833 5/20 0.44
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HTT P42858 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 1/20 0.41
PKM P14618 2/20 0.39
NPC1 O15118 1/20 0.39
MITF O75030 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
EGLN1 Q9GZT9 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
GRM5 P41594 1/20 0.39
HSD17B14 Q9BPX1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6564996 0.91 KMT2A (0.54) KMT2AGRM4ALDH1A1MAPTHPGD
SCHEMBL7670696 0.87 KMT2A (0.44) KMT2AKDM4EPKMNPC1MITF
SCHEMBL6563532 0.84 ALDH1A1 (0.44) KMT2AALDH1A1MAPTHPGDNPSR1
SCHEMBL6565480 0.79 GSK3B (0.47) ALDH1A1SMN1; SMN2VNN1
SCHEMBL6563651 0.79 MAPK13 (0.45) KMT2AALDH1A1HTTMEN1NPC1
SCHEMBL6565285 0.79 NPC1 (0.49) ALDH1A1MAPTNPC1RAB9AEGLN1
SCHEMBL6562338 0.78 GAA (0.47) KMT2AALDH1A1MAPTHTTSMN1; SMN2
SCHEMBL6565408 0.77 CNR1 (0.41) KMT2AALDH1A1MAPTHPGDNPSR1
SCHEMBL7677085 0.76 VNN1 (0.46) EGLN1PTGDR2GRM5VNN1
SCHEMBL6561875 0.76 HPGD (0.47) KMT2AALDH1A1MAPTHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed