SCHEMBL6565408

SCHEMBL6565408

COC(=O)c1ccccc1C(=O)c1ccc(C#CCNc2ccc(C#N)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ALDH1A1 P00352 5/20 0.39
RAB9A P51151 4/20 0.39
NPC1 O15118 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
HPGD P15428 1/20 0.39
AGTR1 P30556 1/20 0.39
GCGR P47871 1/20 0.39
PTPN11 Q06124 1/20 0.38
VNN1 O95497 1/20 0.38
HIF1A Q16665 1/20 0.38
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
LMNA P02545 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563946 0.87 KLK1 (0.42) CA1CA2ALDH1A1RAB9ANPC1
SCHEMBL6563651 0.86 MAPK13 (0.45) CNR1CNR2ALDH1A1RAB9ANPC1
SCHEMBL6563532 0.84 ALDH1A1 (0.44) CNR1CNR2ALDH1A1RAB9ANPC1
SCHEMBL6563213 0.80 KMT2A (0.39) CNR1CNR2RAB9ANPC1VNN1
SCHEMBL6565480 0.79 GSK3B (0.47) CA1CA2ALDH1A1SMN1; SMN2VNN1
SCHEMBL28782860 0.78 CA1 (0.56) CA1CA2ALDH1A1RAB9ANPC1
SCHEMBL6565441 0.77 KMT2A (0.46) ALDH1A1RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL6561875 0.76 HPGD (0.47) ALDH1A1RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL6565256 0.75 AKR1C3 (0.44) ALDH1A1HSD17B10ATM
SCHEMBL6565461 0.75 VNN1 (0.48) VNN1KMT2AMEN1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed
EP-1140802-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM KG (DE) 2001-10-10 EP disclosed
WO-2000035859-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-06-22 WO disclosed