SCHEMBL6565568

SCHEMBL6565568

Cc1ccc(NC(=O)N(Cc2ccccc2)C2=COCO2)c(O)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.45
CXCR2 P25025 1/20 0.44
KMT2A Q03164 3/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
JAK2 O60674 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
PAX8 Q06710 1/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
PTK2 Q05397 1/20 0.37
TSPO P30536 1/20 0.37
UBE2M P61081 2/20 0.36
DCUN1D1 Q96GG9 2/20 0.36
NR1H4 Q96RI1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4355633 0.89 PDK1 (0.43) UBE2MDCUN1D1
SCHEMBL4345516 0.81 ALOX15 (0.48) GAAKMT2AMEN1HTTTP53
SCHEMBL4342089 0.80 ALDH1A1 (0.34) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL4352899 0.80 EGFR (0.41) KMT2AMEN1ALDH1A1HTTUBE2M
SCHEMBL4345577 0.79 HDAC3 (0.36) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL4355478 0.78 EGFR (0.43) NPC1RAB9AALDH1A1HTTUBE2M
SCHEMBL4341341 0.78 RAB9A (0.36) KMT2AMEN1NPC1RAB9AALDH1A1
SCHEMBL4351294 0.78 ALDH1A1 (0.39) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL4359232 0.77 ACHE (0.39) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL4354386 0.77 CCR2 (0.41) GAAKMT2AMEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed