SCHEMBL6572343

SCHEMBL6572343

COCCN(CCOC)c1ccc(N)c(-c2ccccc2C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.40
CYP2C19 P33261 4/20 0.40
CYP3A4 P08684 3/20 0.40
ALOX15 P16050 2/20 0.40
TSHR P16473 2/20 0.40
HSD17B10 Q99714 2/20 0.40
KDM4E B2RXH2 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
CLK4 Q9HAZ1 3/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
GLA P06280 2/20 0.38
CYP2C9 P11712 1/20 0.38
BACE1 P56817 1/20 0.38
TRPA1 O75762 4/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 2/20 0.36
CYP2D6 P10635 1/20 0.36
MAPK1 P28482 1/20 0.36
AR P10275 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572612 0.83 BACE1 (0.40) TSHRKDM4EGLABACE1TRPA1
SCHEMBL6572502 0.83 S100B (0.40) CYP1A2CYP2C19ALOX15HSD17B10KDM4E
SCHEMBL6573203 0.83 ALDH1A1 (0.34) ALOX15HSD17B10TDP1BACE1ALDH1A1
SCHEMBL6571124 0.82 F2 (0.36) KDM4EALDH1A1CRHR1F2PRSS1
SCHEMBL6570863 0.82 CRHR1 (0.39) CYP1A2CYP2C19CYP3A4TDP1CLK4
SCHEMBL6571532 0.82 HTR7 (0.44) CYP1A2CYP2C19CYP3A4HSD17B10TDP1
SCHEMBL6572540 0.80 S100B (0.34) CYP1A2CYP2C19CYP3A4HSD17B10CYP2C9
SCHEMBL6571801 0.79 ALDH1A1 (0.37) ALDH1A1CRHR1F2PRSS1PRSS2
SCHEMBL6571350 0.79 CYP1A2 (0.40) CYP1A2CYP2C19CYP3A4ALOX15TSHR
SCHEMBL6572101 0.78 CRHR1 (0.36) CLK4BACE1CRHR1F2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed