SCHEMBL6576502

SCHEMBL6576502

C#Cc1ccc2ccc(=O)n(-c3ccc(C)cc3)c2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 6/20 0.36
LMNA P02545 2/20 0.35
HTT P42858 2/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSP90AA1 P07900 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
XBP1 P17861 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TLR9 Q9NR96 1/20 0.35
NOTUM Q6P988 1/20 0.35
CYP2C9 P11712 1/20 0.34
CDC7 O00311 1/20 0.34
CDK2 P24941 1/20 0.34
APLNR P35414 1/20 0.34
HTR7 P34969 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578565 0.81 TDP2 (0.35) TDP2LMNAHTTNPC1ALDH1A1
SCHEMBL8040091 0.74 CA12 (0.52) LMNAHTTNPC1ALDH1A1HSP90AA1
SCHEMBL6578645 0.68 HSD11B1 (0.40) HTTALDH1A1RAB9ANPSR1NOTUM
SCHEMBL13444931 0.68 ALDH1A1 (0.59) NPC1ALDH1A1HPGDMAPK1RAB9A
SCHEMBL5922702 0.68 HTR6 (0.48) LMNAHTTALDH1A1MAPTHPGD
SCHEMBL18674301 0.67 POLB (0.36) NPC1MAPTRAB9AKDM4EKMT2A
SCHEMBL13663703 0.66 CYP2A6 (0.59) LMNAALDH1A1HPGDKDM4E
SCHEMBL5014194 0.65 PTGS2 (0.46) HTTALDH1A1MAPTMAPK1RAB9A
SCHEMBL121302 0.64
SCHEMBL18029368 0.64 HTR7 (0.49) MAPTCDC7CDK2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937045-B1 N-ARYL SUBSTITUTED TETRAHYDROQUINOLINES LIGANDS FOR RETINOID RECEPTORS HAVING AGONIST, ANTAGONIST OR INVERSE AGONIST TYPE ACTIVITY ALLERGAN INC (US) 2004-04-28 EP disclosed