SCHEMBL6582104

SCHEMBL6582104

CCOC(=O)Oc1c[nH]nc1NC1CC(C)(c2cccc(Br)c2)OC1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 11/20 0.34
ALDH1A1 P00352 4/20 0.33
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
SLC6A2 P23975 1/20 0.32
CHRNB4 P30926 1/20 0.32
SLC6A4 P31645 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
SLC6A3 Q01959 1/20 0.32
CHRND Q07001 1/20 0.32
HCAR3 P49019 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
CACNA1F O60840 1/20 0.32
ABCB1 P08183 1/20 0.32
CACNA1D Q01668 1/20 0.32
CACNA1S Q13698 1/20 0.32
CACNA1C Q13936 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6288883 0.87 SLC26A6 (0.37) IDO1ALDH1A1CHRNA1CHRNGCHRNB1
SCHEMBL6585426 0.84 HPGDS (0.33) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL6152031 0.84 OPRM1 (0.32)
SCHEMBL6581680 0.79 ALDH1A1 (0.36) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL6581698 0.78 ALDH1A1 (0.32) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL6579675 0.77 TYMS (0.32) ALDH1A1HTTSMN1; SMN2
SCHEMBL6152278 0.71 ALDH1A1 (0.45) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL6291829 0.71 JAK2 (0.40) ALDH1A1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL6152574 0.70 SYK (0.35) KDM4EMEN1KMT2ATDP1CASP1
SCHEMBL5776027 0.69 CHRNA1 (0.35) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406888-A1 SUBSTITUTED $G(G)-LACTONE COMPOUNDS SERVING AS NMDA ANTAGONISTS Grünenthal GmbH (DE) 2004-04-14 EP claimed
WO-2003004483-A1 SUBSTITUTED $G(G)-LACTONE COMPOUNDS SERVING AS NMDA ANTAGONISTS Grünenthal GmbH (DE) 2003-01-16 WO claimed
EP-1406888-A1 SUBSTITUTED $G(G)-LACTONE COMPOUNDS SERVING AS NMDA ANTAGONISTS Grünenthal GmbH (DE) 2004-04-14 EP disclosed
WO-2003004483-A1 SUBSTITUTED $G(G)-LACTONE COMPOUNDS SERVING AS NMDA ANTAGONISTS Grünenthal GmbH (DE) 2003-01-16 WO disclosed