SCHEMBL6637256

SCHEMBL6637256

Cc1ccc(S(=O)(=O)N(c2ccc(OC(=O)N3CCN(C)CC3)cc2)[C@@](C)(C(=O)O)C(=O)[C@H]2NC(C)(C)CS2)cc1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPY2R P49146 4/20 0.38
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAPT P10636 2/20 0.32
MAPK1 P28482 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6633703 0.86 ALDH1A1 (0.37) NPY2RALDH1A1MAPTKEAP1NFE2L2
SCHEMBL6631941 0.80 NPY2R (0.39) NPY2RALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6633768 0.79 TDP1 (0.35) NPY2RALDH1A1MAPT
SCHEMBL6635356 0.78 NPY2R (0.32) NPY2R
SCHEMBL6634428 0.78 ALDH1A1 (0.33) ALDH1A1MAPT
SCHEMBL6638472 0.77 NPY2R (0.40) NPY2RALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL3848898 0.77 ITGB1 (0.38) NPY2RALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6635534 0.76 ALDH1A1 (0.33) ALDH1A1MAPT
SCHEMBL6632994 0.76 HTR1A (0.31)
SCHEMBL6633698 0.76 HSD17B10 (0.38) NPY2RALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000051-B1 CARBAMYLOXY COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2004-05-19 EP claimed