SCHEMBL6633703

SCHEMBL6633703

Cc1ccc(S(=O)(=O)N(c2ccc(OC(=O)N(C)C)cc2)[C@@](C)(C(=O)O)C(=O)[C@H]2NC(C)(C)CS2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
PTGES O14684 1/20 0.36
KDM4E B2RXH2 1/20 0.32
HSP90AA1 P07900 1/20 0.32
MAPT P10636 1/20 0.32
PPARG P37231 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
RAB9A P51151 1/20 0.32
LMNA P02545 2/20 0.32
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.31
POLB P06746 1/20 0.31
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
RXRG P48443 1/20 0.31
NPY2R P49146 1/20 0.30
KEAP1 Q14145 1/20 0.30
NFE2L2 Q16236 1/20 0.30
MCOLN3 Q8TDD5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6633780 0.93 NCEH1 (0.32) RAB9AGAANPY2R
SCHEMBL6633768 0.93 TDP1 (0.35) ALDH1A1KDM4EMAPTRAB9AGAA
SCHEMBL6634428 0.91 ALDH1A1 (0.33) ALDH1A1PTGESKDM4EHSP90AA1MAPT
SCHEMBL6635534 0.90 ALDH1A1 (0.33) ALDH1A1PTGESKDM4EHSP90AA1MAPT
SCHEMBL6635393 0.89 HSD11B1 (0.32)
SCHEMBL6632994 0.86 HTR1A (0.31)
SCHEMBL6633399 0.86 KEAP1 (0.36) ALDH1A1MAPTKMT2AGAAKEAP1
SCHEMBL6637256 0.86 NPY2R (0.38) ALDH1A1MAPTNPY2RKEAP1NFE2L2
SCHEMBL6632832 0.84 NCEH1 (0.31)
SCHEMBL6632840 0.84 TDP1 (0.32) ALDH1A1KDM4EMAPTRAB9AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000051-B1 CARBAMYLOXY COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2004-05-19 EP claimed