SCHEMBL6656572

SCHEMBL6656572

CNC(=S)N(c1ccccc1)C1CCN(C(=O)O)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 6/20 0.45
SIGMAR1 Q99720 2/20 0.45
OPRD1 P41143 8/20 0.45
LMNA P02545 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CHRM3 P20309 4/20 0.43
OPRK1 P41145 3/20 0.43
ADRA1A P35348 2/20 0.43
ADRA1B P35368 2/20 0.43
SLC22A1 O15245 1/20 0.43
NR1I2 O75469 1/20 0.43
ABCB1 P08183 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD2 P14416 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
MAOA P21397 1/20 0.43
DRD4 P21917 1/20 0.43
MAOB P27338 1/20 0.43
HRH1 P35367 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7247490 0.85 MEN1 (0.61)
SCHEMBL6630919 0.78 LMNA (0.47) SIGMAR1LMNAL3MBTL1HRH1SLC6A3
SCHEMBL3630848 0.77 MEN1 (0.48) OPRM1SIGMAR1OPRD1CHRM3OPRK1
SCHEMBL2896994 0.76 L3MBTL3 (0.46) OPRM1SIGMAR1OPRD1CHRM3OPRK1
SCHEMBL18770884 0.74 MITF (0.71) OPRM1SIGMAR1OPRD1LMNACHRM3
SCHEMBL13801291 0.72 OPRM1 (0.45) OPRM1SIGMAR1OPRD1CHRM3OPRK1
SCHEMBL6630325 0.72 MEN1 (0.63)
SCHEMBL18792902 0.70 OPRM1 (0.65) OPRM1SIGMAR1OPRD1CHRM3OPRK1
SCHEMBL5992931 0.70 ALDH1A1 (0.56) OPRM1SIGMAR1LMNAL3MBTL1OPRL1
SCHEMBL5992920 0.70 ALDH1A1 (0.56) OPRM1SIGMAR1LMNAL3MBTL1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1417202-A2 AMINOPIPERIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 2004-05-12 EP disclosed
WO-2002079186-A2 AMINOPIPERIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 2002-10-10 WO disclosed