SCHEMBL6659765

SCHEMBL6659765

COC(=O)C(Cc1ccc(OC(C)=O)c(OC)c1)NC(C)=O

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.53
ALDH1A1 P00352 3/20 0.51
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
LDHA P00338 1/20 0.49
ACACB O00763 1/20 0.47
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
LCK P06239 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TACR1 P25103 2/20 0.45
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6659770 1.00 PTGS1 (0.53) PTGS1ALDH1A1KMT2AMEN1LDHA
SCHEMBL23417656 0.95 ALOX15 (0.49) PTGS1ALDH1A1KMT2AMEN1LCK
SCHEMBL8410630 0.92 LDHA (0.57) ALDH1A1KMT2AMEN1LDHAACACB
SCHEMBL10425937 0.90 LDHA (0.56) PTGS1ALDH1A1KMT2AMEN1LDHA
SCHEMBL9819533 0.90 LDHA (0.56) PTGS1ALDH1A1KMT2AMEN1LDHA
SCHEMBL9405347 0.90 LDHA (0.56) PTGS1ALDH1A1KMT2AMEN1LDHA
SCHEMBL21510392 0.85 TACR1 (0.50) PTGS1ALDH1A1KMT2AMEN1TACR1
SCHEMBL18489065 0.84 TAS1R3 (0.52) ALDH1A1KMT2AMEN1LDHAACACB
SCHEMBL13481269 0.84 ALOX15 (0.46) PTGS1LCK
SCHEMBL1067908 0.84 ALOX15 (0.46) PTGS1KMT2ALCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8227640-B2 Palladium catalysts INSTITUTE OF BIOENGINEERING AND NANOTECHNOLOGY (SG) 2012-07-24 US disclosed
US-8227640-B2 Palladium catalysts INSTITUTE OF BIOENGINEERING AND NANOTECHNOLOGY (SG) 2012-07-24 US disclosed
US-20100113832-A1 PALLADIUM CATALYSTS AGENCY FOR SCIENCE ,TECHNOLOGY AND RESEARCH (SG) 2010-05-06 US disclosed
US-20100113832-A1 PALLADIUM CATALYSTS AGENCY FOR SCIENCE ,TECHNOLOGY AND RESEARCH (SG) 2010-05-06 US disclosed
WO-2008118097-A1 PALLADIUM CATALYSTS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2008-10-02 WO disclosed
EP-1030854-B1 CATALYSTS FOR ASYMMETRIC SYNTHESIS CONTAINING RIGID CHIRAL LIGANDS PENN STATE RES FOUND (US) 2004-08-18 EP disclosed
US-6380416-B2 CHIRAL BIDENTATE PHOSPHINE LIGANDS WITH CYCLIC RINGS TO RESTRICT CONFORMATIONAL FLEXIBILITY OF THE LIGANDS TO ENHANCE EFFICIENCY; STEREOSELECTIVE HYDROGENATION OF KETONES TO ALCOHOLS, AND A-ACETOAMIDOCINNAMIC ACID TO ACYLAMINO ACIDS THE PENN STATE RESEARCH FOUNDATION 2002-04-30 US disclosed
US-20010047113-A1 Chiral bidentate phosphine ligands with cyclic rings to restrict conformational flexibility of the ligands to enhance efficiency; stereoselective hydrogenation of ketones to alcohols, and a-acetoamidocinnamic acid to acylamino acids THE PENN STATE RESEARCH FOUNDATION 2001-11-29 US disclosed
US-6278024-B1 AS CATALYSTS FOR ASSYMETRIC SYNTHESIS THE PENN STATE RESEARCH FOUNDATION 2001-08-21 US disclosed
US-6207868-B1 BASED ON CHIRAL BIDENTATE PHOSPHINE LIGANDS WITH CYCLIC RING STRUCTURES TO RESTRICT CONFORMATIONAL FLEXIBILITY, ASYMMETRIC SYNTHESIS OF ALCOHOLS BY ENANTIOSELECTIVE HYDROGENATION OF KETONES CATALYZED BY THE CHIRAL LIGANDS THE PENN STATE RESEARCH FOUNDATION 2001-03-27 US disclosed
CN-1281460-A Catalysts for asymmetric synthesis containing rigid chiral ligands PENN STATE RES FOUND (US) 2001-01-24 CN disclosed
EP-0498507-A1 Process for the preparation of enantiomers of alpha-amino acid derivatives by asymmetric hydrogenation DSM N.V. (NL) 1992-08-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010047113-A1 Chiral bidentate phosphine ligands with cyclic rings to restrict conformational flexibility of the ligands to enhance efficiency; stereoselective hydrogenation of ketones to alcohols, and a-acetoamidocinnamic acid to acylamino acids ADH1A, AASDHPPT, AADAT PTGS1 2620/4885ALDH1A1 139/4885KMT2A 391/4885
US-20100113832-A1 PALLADIUM CATALYSTS PDCD1LG2, CD274, PDCD6IP PTGS1 1698/4885ALDH1A1 958/4885KMT2A 3328/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.