SCHEMBL6660079

SCHEMBL6660079

COc1ccnc(N2CCN(C(=O)Cc3csc4ccccc34)CC2)n1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 10/20 0.45
HCRTR2 O43614 10/20 0.45
KDM4E B2RXH2 3/20 0.45
HSD17B10 Q99714 3/20 0.45
MAPT P10636 2/20 0.45
LMNA P02545 1/20 0.45
TSHR P16473 1/20 0.45
ALDH1A1 P00352 3/20 0.45
ACHE P22303 2/20 0.43
CXCR3 P49682 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PANK3 Q9H999 1/20 0.41
HPGD P15428 1/20 0.41
HTR1A P08908 1/20 0.41
TSPO P30536 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6655399 0.80 GFER (0.61) HCRTR1HCRTR2KDM4EHSD17B10MAPT
Hydrochloric Acid SCHEMBL6653320 0.79 GFER (0.60) HCRTR1HCRTR2KDM4EHSD17B10MAPT
Hypochlorous Acid SCHEMBL6653323 0.78 GFER (0.59) HCRTR1HCRTR2KDM4EHSD17B10MAPT
Hydrochloric Acid SCHEMBL8151820 0.74 OPRM1 (0.49) KDM4EMAPTLMNATSHRKMT2A
SCHEMBL6655479 0.74 ALDH1A1 (0.74) HCRTR1HCRTR2MAPTLMNAALDH1A1
Hydrochloric Acid SCHEMBL6654568 0.73 ALDH1A1 (0.72) HCRTR1HCRTR2MAPTLMNAALDH1A1
Hypochlorous Acid SCHEMBL6654575 0.73 ALDH1A1 (0.72) HCRTR1HCRTR2MAPTLMNAALDH1A1
SCHEMBL6674771 0.73 L3MBTL1 (0.59) HCRTR1HCRTR2KDM4EHSD17B10TSHR
SCHEMBL6651379 0.73 ACHE (0.53) HCRTR1HCRTR2ACHEMEN1KMT2A
SCHEMBL6653680 0.73 HCRTR1 (0.40) HCRTR1HCRTR2MAPTHTR1ATSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006110-B1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS ESTEVE LABOR DR (ES) 2004-02-11 EP claimed
US-6372746-B1 ANTICONVULSIVE AGENTS, SEDATIVES AND EATING DISORDERS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2002-04-16 US claimed
EP-1006110-A1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2000-06-07 EP claimed