SCHEMBL6662371

SCHEMBL6662371

CN1C(=O)C(Cc2cccc(F)c2)C(=O)c2cc(C(=O)O)ccc21.NC(=O)c1ccncc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.38
PARP10 Q53GL7 1/20 0.38
KDM4C Q9H3R0 2/20 0.38
KDM5A P29375 2/20 0.38
KDM5B Q9UGL1 2/20 0.38
ROCK2 O75116 2/20 0.35
CDC7 O00311 1/20 0.35
MAP4K4 O95819 1/20 0.35
PIM1 P11309 1/20 0.35
CDK2 P24941 1/20 0.35
GSK3B P49841 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
ROCK1 Q13464 1/20 0.35
HTR7 P34969 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6664500 0.90 NR1H2 (0.41) KDM4CKDM5AKDM5BHTR7NR1H2
SCHEMBL6665597 0.90 ROCK2 (0.41) KDM4CKDM5AKDM5BROCK2ROCK1
SCHEMBL6664526 0.89 PARP10 (0.44) MAOBPARP10NR4A2
SCHEMBL6664689 0.89 PSEN1 (0.43) KDM4CKDM5AKDM5BROCK2ROCK1
SCHEMBL6664479 0.86 ROCK2 (0.40) KDM5AKDM5BROCK2ROCK1PSEN1
SCHEMBL6669268 0.86 ROCK2 (0.38) KDM4CKDM5AKDM5BROCK2ROCK1
SCHEMBL6663534 0.85 NNMT (0.41) MAOBPARP10KDM5AKDM5BOPRM1
SCHEMBL6663962 0.85 ROCK2 (0.46) ROCK2ROCK1PSEN1PSEN2APH1B
Niacinamide SCHEMBL6669309 0.80 PSEN1 (0.41) ROCK2HTR7PSEN1PSEN2APH1B
SCHEMBL6678968 0.80 NR1H2 (0.49) KDM4CNR1H2NR1H3PARK7KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed