SCHEMBL6664689

SCHEMBL6664689

CN1C(=O)C(Cc2ccc(F)c(F)c2)C(=O)c2cc(C(=O)O)ccc21.NC(=O)c1ccncc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
ROCK2 O75116 3/20 0.37
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
HTR7 P34969 1/20 0.34
ROCK1 Q13464 1/20 0.34
FYN P06241 1/20 0.34
VNN1 O95497 1/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
CYP17A1 P05093 1/20 0.33
DPP4 P27487 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6664479 0.92 ROCK2 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6669268 0.92 ROCK2 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
Niacinamide SCHEMBL6669309 0.90 PSEN1 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6680077 0.90 NR1H2 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6663962 0.89 ROCK2 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6662371 0.89 MAOB (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6665597 0.87 ROCK2 (0.41) ROCK2KDM5AKDM4CKDM5BROCK1
SCHEMBL6685279 0.81 NR1H2 (0.38) ROCK2KDM5AKDM4CKDM5BNR1H2
SCHEMBL6681227 0.81 PRKAG1 (0.39) ROCK2KDM5AKDM5BNR1H2NR1H3
SCHEMBL6667909 0.78 NNMT (0.40) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed