SCHEMBL6663962

SCHEMBL6663962

CN1C(=O)C(Cc2ccc(Cl)cc2)C(=O)c2cc(C(=O)O)ccc21.NC(=O)c1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 7/20 0.46
ROCK1 Q13464 3/20 0.42
IP6K1 Q92551 1/20 0.38
CCKBR P32239 3/20 0.36
CCKAR P32238 1/20 0.36
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
CYP17A1 P05093 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6664479 0.90 ROCK2 (0.40) ROCK2ROCK1CCKBRCCKARPSEN1
SCHEMBL6665597 0.90 ROCK2 (0.41) ROCK2ROCK1
SCHEMBL6664550 0.89 ROCK2 (0.43) ROCK2ROCK1IP6K1CCKBRCCKAR
SCHEMBL6664689 0.89 PSEN1 (0.43) ROCK2ROCK1CCKBRCCKARPSEN1
SCHEMBL6669268 0.89 ROCK2 (0.38) ROCK2ROCK1PSEN1PSEN2APH1B
SCHEMBL6662371 0.85 MAOB (0.38) ROCK2ROCK1PSEN1PSEN2APH1B
SCHEMBL6665581 0.84 NNMT (0.43) ROCK2
SCHEMBL6678968 0.80 NR1H2 (0.49) CCKBR
SCHEMBL6662847 0.79 TSHR (0.41) ROCK2CCKBR
SCHEMBL6681227 0.79 PRKAG1 (0.39) ROCK2CCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed