SCHEMBL6665597

SCHEMBL6665597

CN1C(=O)C(Cc2cccc(Cl)c2)C(=O)c2cc(C(=O)O)ccc21.NC(=O)c1ccncc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.41
KDM4C Q9H3R0 2/20 0.38
KDM5B Q9UGL1 2/20 0.37
CSNK2A2 P19784 2/20 0.37
ROCK1 Q13464 1/20 0.37
CSNK2B P67870 1/20 0.37
KDM4A O75164 1/20 0.37
PDE5A O76074 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
KDM5A P29375 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
LMNA P02545 1/20 0.35
OPRK1 P41145 1/20 0.35
PDE3A Q14432 1/20 0.35
CSNK2A1 P68400 1/20 0.35
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6663962 0.90 ROCK2 (0.46) ROCK2ROCK1
SCHEMBL6680821 0.90 ALDH1A1 (0.41) KDM4CPDE5AALDH1A1MAPTNR1H2
SCHEMBL6662371 0.90 MAOB (0.38) ROCK2KDM4CKDM5BCSNK2A2ROCK1
SCHEMBL6664479 0.88 ROCK2 (0.40) ROCK2KDM5BROCK1KDM5ANR1H2
SCHEMBL6664689 0.87 PSEN1 (0.43) ROCK2KDM4CKDM5BROCK1ALDH1A1
SCHEMBL6669268 0.86 ROCK2 (0.38) ROCK2KDM4CKDM5BROCK1KDM5A
SCHEMBL6665423 0.85 NNMT (0.41) KDM5BCSNK2A2PDE5AKDM5AOPRK1
SCHEMBL6678968 0.80 NR1H2 (0.49) KDM4CALDH1A1NR1H2NR1H3PARK7
SCHEMBL6664550 0.79 ROCK2 (0.43) ROCK2ROCK1ALDH1A1NR1H2NR1H3
Niacinamide SCHEMBL6669309 0.79 PSEN1 (0.41) ROCK2ALDH1A1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed