SCHEMBL6663236

SCHEMBL6663236

CS(=O)(=O)Nc1ccc(F)cc1Br

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
PTGS2 P35354 5/20 0.44
CA2 P00918 2/20 0.43
CA1 P00915 1/20 0.43
SLC22A12 Q96S37 2/20 0.42
PTGS1 P23219 3/20 0.42
THRB P10828 1/20 0.42
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP19A1 P11511 1/20 0.40
PTGES2 Q9H7Z7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6663333 0.82 PSIP1 (0.50) CA2CA1THRBPTGES2
SCHEMBL10626704 0.81 PTGS2 (0.56) PTGS2PTGS1THRB
SCHEMBL1290883 0.79 KMT2A (0.49) ALDH1A1NPC1MAPTPKMRAB9A
SCHEMBL15108250 0.79 PLA2G7 (0.49) PTGS2SLC22A12PTGS1PKM
SCHEMBL6658979 0.79 CA2 (0.67) PTGS2CA2CA1SLC22A12PTGS1
SCHEMBL16492686 0.78 KMT2A (0.55) PTGS2CA2CA1SLC22A12PTGS1
SCHEMBL4094789 0.78 PTGS2 (0.44) ALDH1A1PTGS2CA2CA1SLC22A12
SCHEMBL17703732 0.76 NR3C1 (0.43) ALDH1A1PTGS2SLC22A12PTGS1PKM
SCHEMBL6662688 0.76 KEAP1 (0.57) CA2CA1
SCHEMBL1688371 0.76 PLA2G7 (0.49) PTGS2SLC22A12PTGS1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244615-B1 METHOD FOR PRODUCING N-SUBSTITUTED 2,4-DIAMINO-5-FLUORO BENZONITRILES AND NOVEL INTERMEDIATES BAYER CROPSCIENCE AG (DE) 2004-08-11 EP disclosed
US-20030017948-A1 Method for producing n-substituted 2,4-diamino-5-fluoro benzonitriles and novel intermediates BAYER AKTIENGESELLSCHAFT (DE) 2003-01-23 US disclosed
EP-1244615-A1 METHOD FOR PRODUCING N-SUBSTITUTED 2,4-DIAMINO-5-FLUORO BENZONITRILES AND NOVEL INTERMEDIATES Bayer Aktiengesellschaft (DE) 2002-10-02 EP disclosed
WO-2001047873-A1 METHOD FOR PRODUCING N-SUBSTITUTED 2,4-DIAMINO-5-FLUORO BENZONITRILES AND NOVEL INTERMEDIATES BAYER AKTIENGESELLSCHAFT (DE) 2001-07-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030017948-A1 Method for producing n-substituted 2,4-diamino-5-fluoro benzonitriles and novel intermediates DDT, PFAS, DAO ALDH1A1 325/4885PTGS2 3174/4885CA2 1965/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.