SCHEMBL6665022

SCHEMBL6665022

CC(C)C[C@H](NC(=O)CBr)C(=O)N[C@@H](Cc1ccc(C2COCCN2C(=O)O)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.42
CYP3A5 P20815 2/20 0.42
CYP3A7 P24462 2/20 0.42
CYP3A43 Q9HB55 2/20 0.42
REN P00797 3/20 0.41
TMPRSS11D O60235 1/20 0.40
CTRL P40313 1/20 0.40
PSMB10 P40306 3/20 0.40
PSMB2 P49721 3/20 0.40
MMP1 P03956 1/20 0.40
PSMB5 P28074 10/20 0.40
PSMB9 P28065 3/20 0.40
PSMB8 P28062 3/20 0.40
PSMB11 A5LHX3 1/20 0.40
PSMD11 O00231 1/20 0.40
PSMD12 O00232 1/20 0.40
PSMD14 O00487 1/20 0.40
PSMA7 O14818 1/20 0.40
PSMD3 O43242 1/20 0.40
CTSB P07858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665016 0.81 REN (0.41) CYP3A4CYP3A5CYP3A7CYP3A43REN
SCHEMBL6473757 0.80 CACNA1B (0.46) CYP3A4CYP3A5CYP3A7CYP3A43REN
SCHEMBL6666207 0.75 CAPN1 (0.45) RENPSMB10PSMB2PSMB5PSMB9
SCHEMBL7339983 0.70 CTSS (0.59) RENPSMB10PSMB2PSMB5PSMB9
SCHEMBL13296580 0.69 MAPT (0.57) MMP1CTSBPOLBMAPTATM
SCHEMBL21981114 0.68 LY96 (0.53) POLBMAPTNPSR1TDP1
SCHEMBL6479130 0.68 CTSK (0.55) CACNA1B
SCHEMBL7345558 0.67 CACNA1B (0.47) RENPSMB10PSMB2MMP1PSMB5
SCHEMBL7345553 0.67 CACNA1B (0.47) RENPSMB10PSMB2MMP1PSMB5
SCHEMBL29861037 0.67 POLB (0.59) RENMMP1POLBMAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140837-B1 COMPOUNDS USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASES GLAXO GROUP LTD (GB) 2004-08-18 EP disclosed