SCHEMBL6667091

SCHEMBL6667091

NC(=O)c1ccncc1.O=C(O)c1ccc2c(c1)C(=O)CC(=O)N2Cc1ccc(F)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.38
PRKAG1 P54619 4/20 0.38
PRKAB1 Q9Y478 4/20 0.38
PRKAA2 P54646 3/20 0.38
HPGD P15428 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PARK7 Q99497 1/20 0.36
KDM5A P29375 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
POLB P06746 1/20 0.35
HTR7 P34969 1/20 0.35
PRKAA1 Q13131 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6666692 0.92 PRKAG1 (0.45) CTRB1PRKAG1PRKAB1PRKAA2HPGD
SCHEMBL6663006 0.92 PRKAG1 (0.40) CTRB1PRKAG1PRKAB1PRKAA2HPGD
SCHEMBL6670369 0.90 PRKAG1 (0.43) CTRB1PTGDR2PRKAG1PRKAB1PRKAA2
SCHEMBL6663894 0.89 ALDH1A1 (0.45) CTRB1PRKAG1PRKAB1PRKAA2HPGD
SCHEMBL6665669 0.87 CPT2 (0.43) PTGDR2PRKAG1PRKAB1PRKAA2HPGD
SCHEMBL6664683 0.87 KMT2A (0.43) CTRB1PRKAG1PRKAB1PRKAA2HPGD
SCHEMBL6665427 0.84 NNMT (0.43) CTRB1PTGDR2PRKAG1PRKAB1PRKAA2
SCHEMBL6668468 0.79 KDM5A (0.41) CTRB1PTGDR2PRKAG1PRKAB1PRKAA2
SCHEMBL6665535 0.79 KDM5A (0.41) CTRB1PTGDR2PRKAG1PRKAB1PRKAA2
SCHEMBL6668559 0.77 NNMT (0.41) PTGDR2PRKAG1PRKAB1PRKAA2KDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed