SCHEMBL6664683

SCHEMBL6664683

NC(=O)c1ccncc1.O=C(O)c1ccc2c(c1)C(=O)CC(=O)N2Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
MDH2 P40926 2/20 0.40
HSP90B1 P14625 1/20 0.40
TRAP1 Q12931 1/20 0.40
CTRB1 P17538 1/20 0.39
HPGD P15428 1/20 0.39
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
CA12 O43570 1/20 0.38
APAF1 O14727 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
BCHE P06276 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6663006 0.92 PRKAG1 (0.40) KMT2AMEN1MAPTLMNACTRB1
SCHEMBL6666692 0.92 PRKAG1 (0.45) KMT2AMEN1MAPTLMNACTRB1
SCHEMBL6670369 0.92 PRKAG1 (0.43) KMT2AMEN1MAPTLMNACTRB1
SCHEMBL6667930 0.89 KMT2A (0.51) KMT2AMEN1MAPTLMNAMDH2
SCHEMBL6665669 0.89 CPT2 (0.43) KMT2AMEN1HPGDTP53CYP1A2
SCHEMBL6667091 0.87 CTRB1 (0.39) KMT2AMEN1CTRB1HPGDCA1
SCHEMBL6663894 0.85 ALDH1A1 (0.45) KMT2AMEN1CTRB1HPGDCA1
SCHEMBL6668468 0.79 KDM5A (0.41) CTRB1TP53PRKAG1PRKAA2PRKAB1
SCHEMBL6665535 0.79 KDM5A (0.41) CTRB1PRKAG1PRKAA2PRKAB1
SCHEMBL6665674 0.78 P2RX3 (0.40) KMT2AMEN1MAPTCTRB1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed