SCHEMBL6663894

SCHEMBL6663894

NC(=O)c1ccncc1.O=C(O)c1ccc2c(c1)C(=O)CC(=O)N2Cc1cccc(F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
KDM4C Q9H3R0 2/20 0.43
NLRP3 Q96P20 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
MAOB P27338 1/20 0.40
PARP10 Q53GL7 1/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
KDM5A P29375 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
PRKAG1 P54619 2/20 0.39
PRKAA2 P54646 2/20 0.39
PRKAB1 Q9Y478 2/20 0.39
CTRB1 P17538 1/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665669 0.89 CPT2 (0.43) KDM4EKMT2AMEN1PRKAG1PRKAA2
SCHEMBL6667091 0.89 CTRB1 (0.39) ALDH1A1KDM4CCA1CA2CA9
SCHEMBL6666774 0.87 MAPT (0.47) ALDH1A1KDM4ECA2CA9MAOB
SCHEMBL6663006 0.86 PRKAG1 (0.40) ALDH1A1CA1CA2CA9KMT2A
SCHEMBL6666692 0.86 PRKAG1 (0.45) CA1CA2CA9KMT2AMEN1
SCHEMBL6666674 0.86 KDM4C (0.42) ALDH1A1KDM4EKDM4CNLRP3MAOB
SCHEMBL6670369 0.86 PRKAG1 (0.43) ALDH1A1CA1CA2CA9KMT2A
SCHEMBL6664683 0.85 KMT2A (0.43) ALDH1A1CA1CA2CA9KMT2A
SCHEMBL6665722 0.84 NNMT (0.43) ALDH1A1KDM4EKDM4CNLRP3MAOB
SCHEMBL6662371 0.76 MAOB (0.38) KDM4CMAOBPARP10KMT2AKDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed