SCHEMBL6674836

SCHEMBL6674836

CCOc1ccc(N(CC)C(N)=NC(=O)OC(C)(C)C)cc1CNC(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4A O75164 1/20 0.33
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
PPARD Q03181 2/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
POLB P06746 1/20 0.32
KCNA5 P22460 1/20 0.31
MEN1 O00255 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
PTPN1 P18031 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678687 0.91 KDM4E (0.38) KDM4ENPC1MAPTRAB9AALDH1A1
SCHEMBL6680479 0.89 CYP2C9 (0.39) KMT2APPARDPPARGMEN1OPRK1
SCHEMBL6676958 0.87 KDM4E (0.36) KDM4ENPC1MAPTRAB9AL3MBTL1
SCHEMBL6677105 0.80 KDM4A (0.36) KDM4ENPC1MAPTRAB9AKMT2A
SCHEMBL8771555 0.78 IDO1 (0.39) KDM4ENPC1MAPTRAB9ACA1
SCHEMBL6687614 0.77 IDO1 (0.41) KDM4ENPC1MAPTRAB9AKMT2A
SCHEMBL6681075 0.77 NQO2 (0.39) KDM4ENPC1MAPTRAB9AKMT2A
SCHEMBL6675899 0.77 KDM4E (0.37) KDM4ENPC1MAPTRAB9AKMT2A
SCHEMBL6681092 0.77 ALDH1A1 (0.42) KDM4EMAPTKMT2AALDH1A1CYP2D6
SCHEMBL6676118 0.76 CA2 (0.47) KDM4ENPC1MAPTRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed