SCHEMBL6676280

SCHEMBL6676280

CC(c1cccc(NC(N)=N[N+](=O)[O-])c1)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
MTOR P42345 1/20 0.37
AURKA O14965 3/20 0.36
RPS6KB1 P23443 3/20 0.36
BACE1 P56817 3/20 0.36
ALDH1A1 P00352 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
AAK1 Q2M2I8 1/20 0.35
CA2 P00918 1/20 0.34
NPY5R Q15761 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7243182 0.82 AURKA (0.41) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7239905 0.82 ALDH1A1 (0.46) MTORAURKARPS6KB1BACE1ALDH1A1
SCHEMBL6676274 0.80 CA2 (0.41) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6547640 0.79 PPARG (0.39) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6679019 0.78 HDAC4 (0.39) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6675007 0.78 GRIN2D (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
Hydrochloric Acid SCHEMBL6679173 0.77 SIGMAR1 (0.48) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6675145 0.76 KMT2A (0.47) AURKARPS6KB1ALDH1A1MEN1KMT2A
SCHEMBL6676180 0.76 SIGMAR1 (0.47) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6681977 0.75 AKT1 (0.43) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed