SCHEMBL6679019

SCHEMBL6679019

CCC(NC(=O)OC(C)(C)C)c1cccc(NC(N)=N[N+](=O)[O-])c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.39
HDAC1 Q13547 2/20 0.39
IDO1 P14902 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGB1 P05556 1/20 0.36
ITGAV P06756 1/20 0.36
ITGA2B P08514 1/20 0.36
ITGB5 P18084 1/20 0.36
CTSK P43235 2/20 0.36
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7243182 0.87 AURKA (0.41) HDAC4HDAC1HDAC3HDAC7HDAC2
SCHEMBL6547640 0.85 PPARG (0.39) HDAC4HDAC1HDAC3HDAC7HDAC2
SCHEMBL6676274 0.82 CA2 (0.41) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6680765 0.82 ALDH1A1 (0.44) HDAC4HDAC1IDO1HDAC3HDAC7
SCHEMBL6679014 0.81 HDAC4 (0.41) HDAC4HDAC1IDO1HDAC3HDAC7
SCHEMBL6676280 0.78 GRIN2D (0.39) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6676599 0.78 MAPT (0.51) MAPTNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL6679740 0.78 AURKA (0.46) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6676387 0.78 SIGMAR1 (0.43) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
Hydrochloric Acid SCHEMBL6676140 0.77 SIGMAR1 (0.42) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6645974-B2 Administering an androstamide compound; osteoporosis, anticancer agents, glandular disorders MERCK & CO., INC. 2003-11-11 US disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed