SCHEMBL6690552

SCHEMBL6690552

N#Cc1cccc(NCCN(C(N)=O)C(=O)[CH]CC2CCCCC2)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.51
KMT2A Q03164 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
CCR3 P51677 5/20 0.37
HTR2A P28223 3/20 0.37
CCR2 P41597 1/20 0.37
EPHX1 P07099 1/20 0.37
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSK P43235 1/20 0.37
CYP2D6 P10635 1/20 0.36
OPRK1 P41145 1/20 0.36
GRM5 P41594 1/20 0.36
SYK P43405 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687814 0.88 EPHX1 (0.40) TSHRKMT2ACCR2EPHX1CYP2D6
SCHEMBL6693491 0.86 NPC1 (0.42) KMT2AL3MBTL1
SCHEMBL6688042 0.85 HTR7 (0.39) KMT2AOPRK1
SCHEMBL6685681 0.85 EPHX2 (0.48) TSHRKMT2AL3MBTL1EPHX1CYP2D6
SCHEMBL6688679 0.83 NPC1 (0.39) KMT2AL3MBTL1EPHX1
SCHEMBL6686695 0.82 MEN1 (0.40) KMT2ACCR3CTSLCTSK
SCHEMBL6686627 0.82 NPC1 (0.38) KMT2ASYK
SCHEMBL6689992 0.81 CFD (0.41) EPHX1
SCHEMBL6687208 0.79 TRPA1 (0.35) KMT2AL3MBTL1EPHX1CYP2D6
SCHEMBL6693494 0.79 SLC6A9 (0.37) EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed