SCHEMBL6687208

SCHEMBL6687208

NC(=O)N(CCNc1c(F)cccc1F)C(=O)[CH]CC1CCCCC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 3/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
CD38 P28907 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
EPHX1 P07099 1/20 0.33
PDE4D Q08499 2/20 0.32
PARP10 Q53GL7 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
ALDH1A1 P00352 2/20 0.31
OPRL1 P41146 1/20 0.31
ALOX5 P09917 1/20 0.31
MEN1 O00255 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6693491 0.85 NPC1 (0.42) TDP1L3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL6685923 0.84 RAB9A (0.38) EPHX1
SCHEMBL6686989 0.82 BTK (0.35) CD38L3MBTL1ALDH1A1OPRL1
SCHEMBL6693494 0.82 SLC6A9 (0.37) EPHX1PARP10ALOX5
SCHEMBL6685915 0.82 RAB9A (0.35) PARP10ALDH1A1OPRL1MEN1KMT2A
SCHEMBL6688042 0.82 HTR7 (0.39) TDP1PARP10ALDH1A1MEN1CYP3A4
SCHEMBL6685681 0.82 EPHX2 (0.48) EPHX1L3MBTL1ALDH1A1MEN1CYP3A4
SCHEMBL6686689 0.81 ALDH1A1 (0.36) EPHX1PARP10L3MBTL1ALDH1A1OPRL1
SCHEMBL6688679 0.80 NPC1 (0.39) TDP1EPHX1L3MBTL1ALDH1A1MEN1
SCHEMBL6690552 0.79 TSHR (0.51) EPHX1L3MBTL1CYP2D6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed