SCHEMBL669124

SCHEMBL669124

Cc1csc(OC(N)=O)c1C

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
GAA P10253 1/20 0.32
POLB P06746 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11798736 0.77 ALDH1A1 (0.34) GAA
SCHEMBL3137968 0.76 ELANE (0.36) KMT2A
SCHEMBL114172 0.72 ADRA2A (0.34) ADRA2AADRA2BADRA2CMEN1KMT2A
SCHEMBL1158351 0.72 ALOX5 (0.42) MEN1KMT2AGAAPOLB
SCHEMBL28583999 0.69 ADRA2A (0.33) ADRA2AADRA2BADRA2CMEN1KMT2A
SCHEMBL9510309 0.69
SCHEMBL27494475 0.68 GAA (0.42) ADRA2AADRA2BADRA2CKMT2AGAA
SCHEMBL28054801 0.67 LMNA (0.35) MEN1KMT2APOLB
SCHEMBL27374876 0.67 LMNA (0.35) ADRA2AADRA2BADRA2CMEN1KMT2A
SCHEMBL28578552 0.65 ALOX15 (0.34) ADRA2AADRA2BADRA2CMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 99 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024119140-A1 CLEAVABLE COMONOMER STRATEGY FOR ACCELERATING REMOVAL OF GEL NAIL POLISH MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2024-06-06 WO disclosed
EP-4359380-A1 PROCESSES FOR THE PREPARATION OF (S)-2-(2,6-DIOXOPIPERIDIN-3-YL)-4-((2-FLUORO-4-((3-MORPHOLINOAZETIDIN-1-YL) METHYL)BENZYL) AMINO)ISOINDOLINE-1,3-DIONE Celgene Corporation (US) 2024-05-01 EP disclosed
WO-2024073745-A1 INHIBITORS OF EGFR OR HER2 AND METHODS OF USE ARBELLA THERAPEUTICS, LLC (US) 2024-04-04 WO disclosed
WO-2023220737-A2 OLIGONUCLEOTIDES HAVING A SYNTHETIC BACKBONE AND SYNTHESIS THEREOF ADARX PHARMACEUTICALS, INC. (US) 2023-11-16 WO disclosed
WO-2023201005-A2 HYDROPHOBIC POLYMER AEROGELS AEROGEL TECHNOLOGIES, LLC (US) 2023-10-19 WO disclosed
WO-2023196342-A1 α4β1/7 INTEGRIN LIGAND CONJUGATED COMPOUNDS AND USES THEREOF ADARX PHARMACEUTICALS, INC. (US) 2023-10-12 WO disclosed
WO-2023146892-A1 BIPHENYL-SUBSTITUTED EPITHELIAL SODIUM CHANNEL BLOCKING COMPOUNDS PARION SCIENCES, INC. (US) 2023-08-03 WO disclosed
WO-2023146896-A1 BICYCLIC-SUBSTITUTED EPITHELIAL SODIUM CHANNEL BLOCKING COMPOUNDS PARION SCIENCES, INC. (US) 2023-08-03 WO disclosed
WO-2023064345-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2023-04-20 WO disclosed
EP-4161651-A1 QUINAZOLINE-DERIVED HCK INHIBITORS FOR USE IN THE TREATMENT OF MYD88 MUTATED DISEASES Dana-Farber Cancer Institute, Inc. (US) 2023-04-12 EP disclosed
EP-2367798-A2 TREATMENT OF AMYOTROPHIC LATERAL SCLEROSIS Cambria Pharmaceuticals, Inc. (US) 2011-09-28 EP disclosed
EP-2337522-A1 ESOPHAGEAL VALVE Vysera Biomedical Limited (IE) 2011-06-29 EP disclosed
WO-2011073970-A1 A GASTROINTESTINAL IMPLANT DEVICE VYSERA BIOMEDICAL LIMITED (IE) 2011-06-23 WO disclosed
EP-2331525-A2 HALOFUGINONE ANALOGS FOR INHIBITION OF TRNA SYNTHETASES AND USES THEREOF President and Fellows of Harvard College (US) 2011-06-15 EP disclosed
WO-2010057006-A9 AZAQUINOLINONE DERIVATIVES AND USES THEREOF LINK MEDICINE CORPORATION (US) 2010-09-16 WO disclosed
WO-2010062372-A2 METHODS FOR MODULATING NF-KB USING GIBBERELLINS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-06-03 WO disclosed
WO-2010059241-A2 TREATMENT OF AMYOTROPHIC LATERAL SCLEROSIS CAMBRIA PHARMACEUTICALS, INC. (US) 2010-05-27 WO disclosed
WO-2010057006-A1 AZAQUINOLINONE DERIVATIVES AND USES THEREOF LINK MEDICINE CORPORATION (US) 2010-05-20 WO disclosed
WO-2010019210-A2 HALOFUGINONE ANALOGS FOR INHIBITION OF TRNA SYNTHETASES AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-02-18 WO disclosed
WO-2009153771-A1 ESOPHAGEAL VALVE VYSERA BIOMEDICAL LIMITED (IE) 2009-12-23 WO disclosed