SCHEMBL6700621

SCHEMBL6700621

O=C(O)c1cc2c([nH]1)N=CN(Cc1ccc(F)c(F)c1)C2

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
CLPP Q16740 3/20 0.37
TSHR P16473 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
RHEB Q15382 1/20 0.37
KDM5A P29375 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
HTT P42858 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
NTRK1 P04629 1/20 0.35
P2RY14 Q15391 1/20 0.34
TBXAS1 P24557 2/20 0.34
PTGER4 P35408 1/20 0.34
TP53 P04637 1/20 0.33
MMP13 P45452 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6704242 0.77 PTGER4 (0.36) ALDH1A1CLPPTSHRL3MBTL1KDM5A
SCHEMBL6700350 0.75 ALDH1A1 (0.32) ALDH1A1CLPPHTT
SCHEMBL6704368 0.74 ALDH1A1 (0.35) ALDH1A1CLPPTSHRL3MBTL1HTT
SCHEMBL6702598 0.71 SIGMAR1 (0.36) ALDH1A1TSHRL3MBTL1HTTSIGMAR1
SCHEMBL30587480 0.62 KDM4C (0.47) KDM5AKDM5BP2RY14MMP13
SCHEMBL18365944 0.62 KDM4C (0.47) KDM5AKDM5BP2RY14MMP13
SCHEMBL8340646 0.61 PTGS1 (0.41) MMP13
SCHEMBL28128191 0.61 GRM2 (0.39) ALDH1A1SIGMAR1PTGER4
SCHEMBL6289350 0.60 KDM5A (0.45) ALDH1A1TSHRRHEBKDM5AKDM5B
SCHEMBL30587615 0.60 CACNA1G (0.59) P2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014916-A1 PYRIMIDINE FUSED BICYCLIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed
US-20040038994-A1 Pyrimidine fused bicyclic metalloproteinase inhibitors WILSON MICHAEL WILLIAM (US) 2004-02-26 US disclosed
WO-2004014916-A1 PYRIMIDINE FUSED BICYCLIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040038994-A1 Pyrimidine fused bicyclic metalloproteinase inhibitors MMP9, MMP1, MMP2 ALDH1A1 221/4885CLPP 3282/4885TSHR 4387/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.