SCHEMBL670494

SCHEMBL670494

COC(=O)C1CC(N)CN1C(=O)OC(C)(C)C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 4/20 0.65
MMP2 P08253 4/20 0.65
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
NR1H2 P55055 2/20 0.41
NR1H3 Q13133 1/20 0.41
PTPN1 P18031 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HTRA1 Q92743 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
P2RX3 P56373 1/20 0.35
PEPD P12955 2/20 0.35
PDE4B Q07343 1/20 0.35
HSD17B10 Q99714 1/20 0.35
XPNPEP1 Q9NQW7 1/20 0.34
MMP1 P03956 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL670493 1.00 ANPEP (0.65) ANPEPMMP2CYP1A2POLBCYP3A4
SCHEMBL2328122 1.00 ANPEP (0.65) ANPEPMMP2CYP1A2POLBCYP3A4
SCHEMBL489156 1.00 ANPEP (0.65) ANPEPMMP2CYP1A2POLBCYP3A4
SCHEMBL1267438 1.00 ANPEP (0.65) ANPEPMMP2CYP1A2POLBCYP3A4
SCHEMBL1267008 1.00 ANPEP (0.65) ANPEPMMP2CYP1A2POLBCYP3A4
SCHEMBL25181712 1.00 ANPEP (0.65) ANPEPMMP2CYP1A2POLBCYP3A4
SCHEMBL1545946 1.00 ANPEP (0.65) ANPEPMMP2CYP1A2POLBCYP3A4
SCHEMBL7729511 1.00 ANPEP (0.65) ANPEPMMP2CYP1A2POLBCYP3A4
Hydrochloric Acid SCHEMBL1412084 0.98 ANPEP (0.63) ANPEPMMP2CYP1A2POLBCYP3A4
Hydrochloric Acid SCHEMBL2347422 0.98 ANPEP (0.63) ANPEPMMP2CYP1A2POLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 70 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250340548-A1 KRAS G12C INHIBITORS FRONTIER MEDICINES CORP (US) 2025-11-06 US disclosed
US-12358886-B2 Heterocyclic compounds for use in the treatment of cancer ARTIOS PHARMA LIMITED (GB) 2025-07-15 US disclosed
US-12291539-B2 KRAS G12C inhibitors FRONTIER MEDICINES CORPORATION (US) 2025-05-06 US disclosed
CN-119395192-B Method for measuring isomers in carfilzomib and preparation thereof by reversed phase liquid chromatography 合肥亿帆生物制药有限公司 2025-04-18 CN disclosed
CN-119395192-A Method for measuring isomers in carfilzomib and preparation thereof by reversed phase liquid chromatography 合肥亿帆生物制药有限公司 2025-02-07 CN disclosed
US-20250019387-A1 KRAS G12C INHIBITORS FRONTIER MEDICINES CORPORATION 2025-01-16 US disclosed
US-20240317748-A1 CARBONYL SUBSTITUTED DIAZASPIRO COMPOUNDS AND ITS USE BIONOVA PHARMACEUTICALS LTD. (KY) 2024-09-26 US disclosed
EP-4426695-A1 KRAS G12C INHIBITORS Frontier Medicines Corporation (US) 2024-09-11 EP disclosed
CN-116888110-A Melanocortin-4 receptor agonists 株式会社LG 化学 2023-10-13 CN disclosed
EP-4010080-B1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER ARTIOS PHARMA LTD (GB) 2023-09-27 EP disclosed
US-7479495-B2 N-heterocyclic inhibitors of TNF-α expression PHARMACOPEIA, INC. (US) 2009-01-20 US disclosed
WO-2008148689-A1 PROLINAMIDE DERIVATIVES AS NK3 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-12-11 WO disclosed
US-20080306086-A1 PROLINAMIDE DERIVATIVES AS NK3 ANTAGONISTS HOFFMANN-LA ROCHE, INC. 2008-12-11 US disclosed
US-20080200535-A1 sphingosine 1-phosphate-1/EDG-1 receptor agonists; autoimmune diseases; immunosuppressants by inducing lymphocyte sequestration in secondary lymphoid tissues; 4-aminocyclopentane-2-encarboxylic acid hydrochloric acid salt ASAHI KASEI PHARMA CORPORATION (JP) 2008-08-21 US disclosed
WO-2008077555-A2 SUBSTITUTED ISOQUINOLINES AND THEIR USE AS RHO-KINASE INHIBITORS SANOFI-AVENTIS (FR) 2008-07-03 WO disclosed
US-20050239770-A1 N-heterocyclic inhibitors of TNF-alpha expression MORIARTY KEVIN J 2005-10-27 US disclosed
US-6906067-B2 N-heterocyclic inhibitors of TNF-α expression BRISTOL-MYERS SQUIBB COMPANY (US) 2005-06-14 US disclosed
WO-2005011697-A2 SULFONAMIDE DERIVATIVES WITH ACTIVITY ON PROTEIN KINASE A AND B ASTEX THERAPEUTICS LIMITED (GB) 2005-02-10 WO disclosed
US-20020137747-A1 N- heterocyclic inhibitors of TNF-alpha expression PHARMACEOPEIA, INC. 2002-09-26 US disclosed
US-20020065270-A1 N-heterocyclic inhibitors of TNF-alpha expression PHARMACOPEIA, INC. 2002-05-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050239770-A1 N-heterocyclic inhibitors of TNF-alpha expression TNF, RELA, NFKBIA ANPEP 1212/4885MMP2 1074/4885CYP1A2 403/4885
US-20240317748-A1 CARBONYL SUBSTITUTED DIAZASPIRO COMPOUNDS AND ITS USE SDHA, PDHA1, GLS ANPEP 1608/4885MMP2 3660/4885CYP1A2 137/4885
US-20080200535-A1 sphingosine 1-phosphate-1/EDG-1 receptor agonists; autoimmune diseases; immunosuppressants by inducing lymphocyte sequestration in secondary lymphoid tissues; 4-aminocyclopentane-2-encarboxylic acid hydrochloric acid salt S1PR1, S1PR2, S1PR4 ANPEP 4289/4885MMP2 4616/4885CYP1A2 2532/4885
US-20020137747-A1 N- heterocyclic inhibitors of TNF-alpha expression TNF, NFKBIA, RELA ANPEP 1460/4885MMP2 1120/4885CYP1A2 315/4885
US-20020065270-A1 N-heterocyclic inhibitors of TNF-alpha expression TNF, NFKBIA, RELA ANPEP 1460/4885MMP2 1120/4885CYP1A2 315/4885
US-12291539-B2 KRAS G12C inhibitors KRAS, NRAS, HRAS ANPEP 4001/4885MMP2 2455/4885CYP1A2 4759/4885
US-20250340548-A1 KRAS G12C INHIBITORS KRAS, NRAS, HRAS ANPEP 4001/4885MMP2 2455/4885CYP1A2 4759/4885
US-20080306086-A1 PROLINAMIDE DERIVATIVES AS NK3 ANTAGONISTS SLC6A3, OPRL1, OPRK1 ANPEP 271/4885MMP2 3631/4885CYP1A2 1733/4885
US-20250019387-A1 KRAS G12C INHIBITORS KRAS, NRAS, HRAS ANPEP 4001/4885MMP2 2455/4885CYP1A2 4759/4885
US-12358886-B2 Heterocyclic compounds for use in the treatment of cancer SDHA, DPYD, TP53 ANPEP 1431/4885MMP2 2027/4885CYP1A2 104/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.