Robenidine

Robenidine

SCHEMBL6729906

N=C(NN=Cc1ccc(Cl)cc1)NN=Cc1ccc(Cl)cc1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
MAPT P10636 4/20 0.50
KMT2A Q03164 4/20 0.49
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 2/20 0.49
GAA P10253 2/20 0.49
AGTR1 P30556 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA4 P22748 1/20 0.48
CA9 Q16790 1/20 0.48
MEN1 O00255 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Robenidine SCHEMBL571509 1.00 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4
Robenidine SCHEMBL3851893 0.98 SMN1; SMN2 (0.51) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4
Robenidine SCHEMBL11769699 0.98 SMN1; SMN2 (0.51) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL19449644 0.91 LMNA (0.58) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL11233334 0.91 MEN1 (0.57) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL23874282 0.91 MAPT (0.47) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL11233329 0.91 MEN1 (0.57) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL16224325 0.91 SMN1; SMN2 (0.54) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11768892 0.90 MEN1 (0.56) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11768897 0.90 MEN1 (0.56) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4310541-A WITH A BIS(BENZYLIDENEAMINO)GUANIDINE MERCK & CO., INC. (US) 1982-01-12 US claimed
US-4041160-A N-METHYL-2-PYRROLIDONE, ANTICOCCIDIAL AGENTS ABIC LTD. (IL) 1977-08-09 US claimed
US-3980705-A Purification of robenidine hydrochloride AMERICAN CYANAMID COMPANY (US) 1976-09-14 US claimed
US-20230147129-A1 COMPOUNDS FOR USE IN THE TREATMENT OF SYNUCLEINOPATHIES UNIVERSITAT AUTÒNOMA DE BARCELONA (ES) 2023-05-11 US disclosed
US-11566012-B2 Methods for treating protozoan infections NEOCULI PTY LTD (AU) 2023-01-31 US disclosed
EP-3960729-A1 COMPOUNDS AND METHODS OF TREATING INFECTIONS Neoculi Pty Ltd (AU) 2022-03-02 EP disclosed
EP-2991968-B1 COMPOUNDS AND METHODS OF TREATING INFECTIONS NEOCULI PTY LTD (AU) 2021-11-10 EP disclosed
US-20210009552-A1 METHODS FOR TREATING PROTOZOAN INFECTIONS NEOCULI PTY LTD (AU) 2021-01-14 US disclosed
US-10829468-B2 Methods for treating protozoan infections NEOCULI PTY LTD. (AU) 2020-11-10 US disclosed
US-20200290990-A1 METHODS FOR TREATING PROTOZOAN INFECTIONS NEOCULI PTY LTD (AU) 2020-09-17 US disclosed
US-10752606-B2 Methods for treating protozoan infections NEOCULI PTY LTD. (AU) 2020-08-25 US disclosed
US-20020123649-A1 Process for the preparation of robenidine and salts thereof LONZA AG (CH) 2002-09-05 US disclosed
US-4310541-A WITH A BIS(BENZYLIDENEAMINO)GUANIDINE MERCK & CO., INC. (US) 1982-01-12 US disclosed
US-4041160-A N-METHYL-2-PYRROLIDONE, ANTICOCCIDIAL AGENTS ABIC LTD. (IL) 1977-08-09 US disclosed
US-3992446-A ANTIPROTOZOAL ACTIVITY, PARTICULARLY AGAINST COCCIDIOSIS AND MALARIA AMERICAN CYANAMID COMPANY (US) 1976-11-16 US disclosed
US-3980705-A Purification of robenidine hydrochloride AMERICAN CYANAMID COMPANY (US) 1976-09-14 US disclosed
US-3954996-A BACTERICIDES ABIC LTD. (IL) 1976-05-04 US disclosed
US-3954996-A BACTERICIDES ABIC LTD. (IL) 1976-05-04 US disclosed
US-3950539-A Substituted diaminoguanidines HOECHST AKTIENGESELLSCHAFT (DT) 1976-04-13 US disclosed
US-3941825-A ANTIPROTOZOA INTERMEDIATES AMERICAN CYANAMID COMPANY (US) 1976-03-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11566012-B2 Methods for treating protozoan infections DPM1, ABCB11, PIGS SMN1; SMN2 3002/4885NPC1 282/4885RAB9A 3198/4885
US-20200290990-A1 METHODS FOR TREATING PROTOZOAN INFECTIONS DPM1, ABCB11, PIGS SMN1; SMN2 3002/4885NPC1 282/4885RAB9A 3198/4885
US-20210009552-A1 METHODS FOR TREATING PROTOZOAN INFECTIONS DPM1, ABCB11, PIGS SMN1; SMN2 3002/4885NPC1 282/4885RAB9A 3198/4885
US-20230147129-A1 COMPOUNDS FOR USE IN THE TREATMENT OF SYNUCLEINOPATHIES SNCA, PARK7, PRNP SMN1; SMN2 6/4885NPC1 801/4885RAB9A 364/4885
US-20020123649-A1 Process for the preparation of robenidine and salts thereof ADH1C, ADH1A, DRD4 SMN1; SMN2 4689/4885NPC1 1482/4885RAB9A 511/4885
US-10829468-B2 Methods for treating protozoan infections DPM1, ABCB11, PIGS SMN1; SMN2 3002/4885NPC1 282/4885RAB9A 3198/4885
US-10752606-B2 Methods for treating protozoan infections DPM1, ABCB11, PIGS SMN1; SMN2 3002/4885NPC1 282/4885RAB9A 3198/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.