SCHEMBL6749339

SCHEMBL6749339

COCN1c2cc(C(CC(=O)O)c3ccccn3)ccc2N(C)c2nccnc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 8/20 0.41
CASP1 P29466 1/20 0.38
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CTSA P10619 3/20 0.33
KCNA5 P22460 2/20 0.33
ITGB3 P05106 2/20 0.33
ITGAV P06756 2/20 0.33
BRD4 O60885 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ABCB11 O95342 1/20 0.33
LMNA P02545 1/20 0.33
ESR1 P03372 1/20 0.33
CYP3A4 P08684 1/20 0.33
ADRA2A P08913 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
PDE4A P27815 1/20 0.33
ADRA1A P35348 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6747727 0.85 BRD4 (0.34) ALDH1A1CYP1A2KCNA5BRD4KDM4E
SCHEMBL6749088 0.84 TSHR (0.36) ALDH1A1CYP1A2KDM4EABCB11LMNA
SCHEMBL7162055 0.75 HSD17B14 (0.41) ALDH1A1KDM4ELMNA
SCHEMBL6751843 0.71 L3MBTL1 (0.37) CYP1A2BRD4
SCHEMBL1131686 0.68 ALDH1A1 (0.55) FFAR1CASP1ALDH1A1CYP1A2KCNA5
SCHEMBL6749056 0.68 CA12 (0.38) ALDH1A1KDM4ELMNA
SCHEMBL8464221 0.67 LMNA (0.33) FFAR1LMNAPDE4A
SCHEMBL6750715 0.67 CASP3 (0.36) ALDH1A1BRD4KDM4E
SCHEMBL6750211 0.65 HDAC6 (0.36)
SCHEMBL6226631 0.61 TNF (0.49) FFAR1ALDH1A1CYP1A2KDM4EABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040092737-A1 Benzopiperidine derivatives EISAI CO., LTD. 2004-05-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092737-A1 Benzopiperidine derivatives HLA-DRB1, HRH1, HRH2 FFAR1 778/4885CASP1 711/4885ALDH1A1 145/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.