SCHEMBL6768482

SCHEMBL6768482

Cc1nc(N)c2nc(C)n(CCNC(=O)c3ccc4ccccc4c3)c2c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.47
HTR1A P08908 8/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C19 P33261 2/20 0.46
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
MAPT P10636 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
KMT2A Q03164 2/20 0.43
SLC6A2 P23975 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6779944 0.94 HDAC3 (0.48) IDO1HTR1AHDAC3HDAC4HDAC1
SCHEMBL6774657 0.89 MAPT (0.49) CYP1A2CYP2D6CYP2C19MAPTSMN1; SMN2
SCHEMBL6773842 0.85 SMN1; SMN2 (0.50) CYP1A2CYP2D6CYP2C19MAPTSMN1; SMN2
SCHEMBL6771355 0.85 POLB (0.47) MAPTSMN1; SMN2KMT2AMEN1NPC1
SCHEMBL6773253 0.85 GAA (0.41) MAPTALDH1A1PKMTP53POLB
SCHEMBL6768729 0.84 TLR7 (0.47) CYP1A2CYP2D6CYP2C19MAPTSMN1; SMN2
SCHEMBL6773364 0.83 RXFP1 (0.43) HDAC3HDAC1MAPTNPC1ALDH1A1
SCHEMBL6773218 0.83 MCHR1 (0.47) HDAC3MAPTALDH1A1PKMPOLB
SCHEMBL6780200 0.83 ALDH1A1 (0.50) CYP1A2HDAC3HDAC1MAPTKMT2A
SCHEMBL6773356 0.83 SMN1; SMN2 (0.48) MAPTSMN1; SMN2KMT2AMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6720333-B2 IMMUNE RESPONSE MODIFIERS; CYTOKINE BIOSYNTHESIS; VIRAL AND NEOPLASTIC DISEASES; N-(4-(4-AMINO-6,7-DIMETHYL-1H-IMIDAZO (4,5-C)PYRIDIN-1-YL)BUTYL)BENZAMIDE 3M INNOVATIVE PROPERTIES COMPANY 2004-04-13 US claimed