SCHEMBL6796572

SCHEMBL6796572

COC(=O)C1=C(OS(=O)(=O)c2ccc(C)cc2)c2ccccc2S(=O)(=O)N1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.52
POLB P06746 1/20 0.52
CYP3A4 P08684 3/20 0.47
CYP2C9 P11712 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CYP2C19 P33261 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
ALDH1A1 P00352 1/20 0.47
RECQL P46063 1/20 0.47
HSD11B1 P28845 2/20 0.46
TP53 P04637 2/20 0.41
CAPN1 P07384 1/20 0.40
VDR P11473 1/20 0.40
DHODH Q02127 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
PKM P14618 1/20 0.39
THPO P40225 1/20 0.39
PMP22 Q01453 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6795739 0.83 HSD11B1 (0.49) MAPTPOLBCYP3A4CYP2C9SMN1; SMN2
SCHEMBL9984200 0.81 MAPT (0.56) MAPTPOLBCYP3A4CYP2C9SMN1; SMN2
SCHEMBL7090095 0.80 MAPT (0.42) MAPTPOLBCYP3A4CYP2C9SMN1; SMN2
Iodide SCHEMBL6794705 0.80 MAPT (0.41) MAPTPOLBCYP3A4CYP2C9SMN1; SMN2
SCHEMBL7334969 0.80 HSD11B1 (0.55) MAPTPOLBCYP3A4CYP2C9SMN1; SMN2
SCHEMBL6794794 0.79 CAPN1 (0.57) MAPTPOLBCYP3A4CYP2C9SMN1; SMN2
SCHEMBL6797487 0.76 MAPT (0.57) MAPTPOLBCYP3A4CYP2C9SMN1; SMN2
SCHEMBL6796426 0.74 HSD11B1 (0.73) CYP3A4CYP2C9CYP2C19HSD11B1LMNA
SCHEMBL30218271 0.74 HSD11B1 (0.73) CYP3A4CYP2C9CYP2C19HSD11B1LMNA
SCHEMBL9984079 0.72 MAPT (0.51) MAPTPOLBCYP3A4CYP2C9SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040063696-A1 1,1-dioxo-2h-1,2-benzothiazine-3-carboxamide derivatives,method for preparing same and pharmaceutical compositions comprising same INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2004-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063696-A1 1,1-dioxo-2h-1,2-benzothiazine-3-carboxamide derivatives,method for preparing same and pharmaceutical compositions comprising same ADCY2, ADCY1, HRH2 MAPT 4376/4885POLB 4037/4885CYP3A4 186/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.