SCHEMBL6813612

SCHEMBL6813612

Clc1ccc(CNC(CN2CCCC2)c2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2C19 P33261 2/20 0.50
ATM Q13315 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
NTSR1 P30989 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
OPRK1 P41145 3/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP3A4 P08684 2/20 0.45
OPRM1 P35372 2/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
TSHR P16473 1/20 0.45
HIF1A Q16665 1/20 0.45
SLC22A1 O15245 1/20 0.45
CHRM2 P08172 1/20 0.45
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13077134 0.88 SMN1; SMN2 (0.50) CYP2D6CYP1A2CYP2C19ATMOPRK1
SCHEMBL3245792 0.86 SMN1; SMN2 (0.46) CYP2D6CYP2C19ATMOPRK1ALDH1A1
SCHEMBL11969235 0.83 LMNA (0.53) TDP1OPRK1KDM4EALDH1A1OPRM1
SCHEMBL8091287 0.79 L3MBTL1 (0.57) CYP2D6CYP1A2CYP2C19ATML3MBTL1
SCHEMBL13039125 0.77 PDE8B (0.46) CYP2D6CYP1A2CYP2C19ATMOPRK1
SCHEMBL17765072 0.77 ALDH1A1 (0.45) CYP2D6CYP2C19ATML3MBTL1OPRK1
SCHEMBL10316558 0.77 SIGMAR1 (0.50) ATML3MBTL1KDM4EMEN1KMT2A
SCHEMBL8716789 0.76 POLB (0.49) CYP2D6CYP1A2CYP2C19NTSR1KDM4E
SCHEMBL9130649 0.76 POLB (0.49) CYP2D6CYP1A2CYP2C19NTSR1KDM4E
SCHEMBL3237722 0.76 GAA (0.50) CYP2D6OPRM1CHRM2ADRA2ACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089965-B1 Urea derivatives for pain management ASTRAZENECA AB (SE) 2004-09-15 EP disclosed
US-6777561-B1 MANAGEMENT OF PAIN; PHENYL-UREA COMPOUNDS ASTRAZENECA CANADA INC. (CA) 2004-08-17 US disclosed