SCHEMBL6825993

SCHEMBL6825993

CC(C)NC(=O)c1nc(-c2ccccc2)c(-c2n[nH]c(=O)cc2C(C)C)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA2B P29275 1/20 0.45
ADORA1 P30542 1/20 0.45
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
CASP1 P29466 1/20 0.43
HPGD P15428 1/20 0.39
CYP1A2 P05177 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PTGS1 P23219 2/20 0.37
XIAP P98170 1/20 0.37
PDE2A O00408 3/20 0.36
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
MLLT1 Q03111 1/20 0.35
HPGDS O60760 1/20 0.35
ACR P10323 1/20 0.35
TP53 P04637 1/20 0.35
TACR2 P21452 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6828337 0.91 CHEK1 (0.40) ADORA3ADORA2AADORA2BADORA1HPGD
SCHEMBL6828463 0.88 ADORA3 (0.46) ADORA3ADORA2AADORA2BADORA1ALOX15
SCHEMBL6829284 0.86 MAPK8 (0.43) ADORA2AADORA1HPGDSMN1; SMN2RAB9A
SCHEMBL6828438 0.86 L3MBTL1 (0.43) TSHRSMN1; SMN2PDE2A
SCHEMBL6828786 0.85 HPGDS (0.49) ADORA3HPGDCYP1A2SMN1; SMN2RAB9A
SCHEMBL6830662 0.83 ADORA3 (0.41) ADORA3ADORA2AADORA2BADORA1ALOX15
SCHEMBL6133796 0.82 ADORA2A (0.50) ADORA3ADORA2AADORA2BADORA1ALOX15
SCHEMBL6828357 0.79 ADORA2A (0.51) ADORA3ADORA2AADORA2BADORA1XIAP
SCHEMBL6829256 0.79 HPGD (0.39) ADORA3ADORA2AADORA1HPGDSMN1; SMN2
SCHEMBL6828483 0.79 XIAP (0.44) ADORA3ADORA2AADORA1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441732-A2 THIAZOLE DERIVATIVE AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-04 EP disclosed
WO-2003039451-A2 THIAZOLE PYRIDAZINONES AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-15 WO disclosed