SCHEMBL6829256

SCHEMBL6829256

CC(=O)N(C)c1nc(-c2ccccc2)c(-c2n[nH]c(=O)cc2C(C)C)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.39
PTGS1 P23219 2/20 0.37
XIAP P98170 2/20 0.35
ALDH1A1 P00352 4/20 0.34
HSP90AA1 P07900 1/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
HPGDS O60760 1/20 0.33
ELANE P08246 1/20 0.33
P2RX3 P56373 1/20 0.33
CCNE2 O96020 1/20 0.32
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6828866 0.83 NPSR1 (0.42) HPGDALDH1A1CYP2C9CYP2C19ROCK1
SCHEMBL6828337 0.80 CHEK1 (0.40) HPGDPTGS1XIAPALDH1A1HSP90AA1
SCHEMBL6825993 0.79 ADORA3 (0.45) HPGDPTGS1XIAPALDH1A1HSP90AA1
SCHEMBL8067393 0.78 KMT2A (0.48) HPGDPTGS1XIAPALDH1A1CYP2C9
SCHEMBL6828786 0.77 HPGDS (0.49) HPGDALDH1A1CYP2C9CYP2C19MEN1
SCHEMBL6829284 0.76 MAPK8 (0.43) HPGDMEN1KMT2ACDK2ADORA2A
SCHEMBL6830646 0.76 ADORA2A (0.53) HPGDXIAPALDH1A1MEN1KMT2A
SCHEMBL6828438 0.76 L3MBTL1 (0.43) ROCK2SMN1; SMN2
SCHEMBL6825783 0.76 ADORA1 (0.56) HPGDXIAPALDH1A1MEN1KMT2A
SCHEMBL6828357 0.75 ADORA2A (0.51) XIAPKMT2AADORA3ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441732-A2 THIAZOLE DERIVATIVE AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-04 EP disclosed
WO-2003039451-A2 THIAZOLE PYRIDAZINONES AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-15 WO disclosed