SCHEMBL6828337

SCHEMBL6828337

CNC(=O)c1nc(-c2ccccc2)c(-c2n[nH]c(=O)cc2C(C)C)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.40
RET P07949 1/20 0.40
PDGFRB P09619 1/20 0.40
PIM1 P11309 1/20 0.40
PDGFRA P16234 1/20 0.40
GSK3B P49841 1/20 0.40
RPS6KA3 P51812 1/20 0.40
LIMK1 P53667 1/20 0.40
CDK5 Q00535 1/20 0.40
TYRO3 Q06418 1/20 0.40
MAPK14 Q16539 1/20 0.40
LRRK2 Q5S007 1/20 0.40
AURKB Q96GD4 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
HPGD P15428 4/20 0.40
XIAP P98170 4/20 0.38
PTGS1 P23219 2/20 0.38
ALDH1A1 P00352 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6825993 0.91 ADORA3 (0.45) HPGDXIAPPTGS1ALDH1A1RAB9A
SCHEMBL6828438 0.87 L3MBTL1 (0.43) RETGSK3BAURKBCLK4HSD17B10
SCHEMBL6829284 0.87 MAPK8 (0.43) PIM1RPS6KA3AURKBCLK4HPGD
SCHEMBL6828786 0.84 HPGDS (0.49) HPGDALDH1A1KDM4EMAPTHSD17B10
SCHEMBL6828357 0.80 ADORA2A (0.51) XIAPNPSR1MAPTHTTRAB9A
SCHEMBL6829256 0.80 HPGD (0.39) HPGDXIAPPTGS1ALDH1A1KDM4E
SCHEMBL6830337 0.79 ADORA2A (0.50) XIAPALDH1A1KDM4ERAB9AADORA3
SCHEMBL6826020 0.79 NPC1 (0.48) HPGDXIAPALDH1A1NPSR1KDM4E
SCHEMBL6828483 0.79 XIAP (0.44) HPGDXIAPALDH1A1NPSR1KDM4E
SCHEMBL6830646 0.79 ADORA2A (0.53) GSK3BHPGDXIAPALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441732-A2 THIAZOLE DERIVATIVE AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-04 EP disclosed
WO-2003039451-A2 THIAZOLE PYRIDAZINONES AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-15 WO disclosed