SCHEMBL6918536

SCHEMBL6918536

CC(C)Cc1nc(-c2ccccn2)oc1C(=O)[C@H](CCc1ccccc1)NC(=O)CCC1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BMP1 P13497 1/20 0.40
KMT2A Q03164 3/20 0.39
HPGD P15428 2/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.37
THRB P10828 1/20 0.37
KCNQ3 O43525 1/20 0.35
KCNQ2 O43526 1/20 0.35
ENPP2 Q13822 1/20 0.35
REN P00797 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
FAAH O00519 4/20 0.35
CES1 P23141 4/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
NCEH1 Q6PIU2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6918530 0.87 BMP1 (0.34) BMP1HPGDALDH1A1KDM4ETHRB
SCHEMBL6918534 0.87 BMP1 (0.34) BMP1HPGDALDH1A1KDM4ETHRB
SCHEMBL7250425 0.80 MMP1 (0.34) BMP1HPGDALDH1A1KDM4ETHRB
SCHEMBL6801151 0.79 CTSL (0.39) RENCTSLCTSBCTSSCTSK
SCHEMBL6799441 0.78 MEN1 (0.41) BMP1KMT2AHPGDMEN1ALDH1A1
SCHEMBL6806942 0.76 CTSL (0.43) RENCTSLCTSBCTSSCTSK
SCHEMBL6463419 0.74 CTSS (0.48) KMT2AMEN1FAAHCES1CTSL
SCHEMBL6465141 0.74 CTSS (0.48) KMT2AMEN1FAAHCES1CTSL
SCHEMBL6468629 0.74 CTSS (0.48) KMT2AMEN1FAAHCES1CTSL
SCHEMBL6472183 0.73 FAAH (0.48) KMT2AHPGDMEN1ALDH1A1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6730671-B2 ENZYME INHIBITOR TREATING AUTOIMMUNE DISEASES, ALZHEIMER'S DISEASE, ATHEROSCLEROSIS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2004-05-04 US disclosed