SCHEMBL6918550

SCHEMBL6918550

CCNS(=O)(=O)c1c[nH]c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.47
HTR2A P28223 1/20 0.45
MEN1 O00255 1/20 0.45
TP53 P04637 1/20 0.45
KMT2A Q03164 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
PKM P14618 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
NR3C1 P04150 2/20 0.43
MGAM O43451 1/20 0.43
TSHR P16473 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1354949 0.84 ALOX12 (0.58) CYP19A1MEN1TP53KMT2ATSHR
SCHEMBL6915427 0.81 FEN1 (0.47) CYP19A1HTR2AMEN1KMT2APKM
SCHEMBL30897273 0.80 ALDH1A1 (0.54) MEN1TP53KMT2ARXFP1PKM
SCHEMBL15416652 0.80 ALDH1A1 (0.54) MEN1TP53KMT2ARXFP1PKM
SCHEMBL9426286 0.79 NSD2 (0.47) CYP19A1MEN1KMT2APKMALDH1A1
SCHEMBL20163593 0.78 CYP19A1 (0.50) CYP19A1ALDH1A1NR3C1MGAM
SCHEMBL19559085 0.78 GPR84 (0.49) HTR2AMEN1TP53KMT2ARXFP1
SCHEMBL6923053 0.76 PBRM1 (0.50) MEN1KMT2APKMALDH1A1TSHR
SCHEMBL29557960 0.75 PBRM1 (0.52) MEN1TP53KMT2ARXFP1PKM
SCHEMBL15415994 0.75 PBRM1 (0.52) MEN1TP53KMT2ARXFP1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040122076-A1 Sulphonamides for the treatment of central nervous system diseases BAYER AKTIENGESELLSCHAFT (DE) 2004-06-24 US disclosed
EP-1335720-A1 SULPHONAMIDES FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISEASES Bayer Aktiengesellschaft (DE) 2003-08-20 EP disclosed
US-6498183-B1 TREATMENT AND PROPHYLAXIS OF DISORDERS CAUSED BY HERPES VIRUSES, IN PARTICULAR HUMAN CYTOMEGALOVIRUS BAYER AKTIENGESELLSCHAFT (DE) 2002-12-24 US disclosed
WO-2002036115-A1 SULPHONAMIDES FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2002-05-10 WO disclosed
EP-1177171-A1 SUBSTITUTED INDOLE SULFONAMIDES AS ANTIVIRAL AGENTS Bayer Aktiengesellschaft (DE) 2002-02-06 EP disclosed
WO-2000066553-A1 SUBSTITUTED INDOLE SULFONAMIDES AS ANTIVIRAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2000-11-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122076-A1 Sulphonamides for the treatment of central nervous system diseases HTR6, SLC6A4, AANAT CYP19A1 3120/4885HTR2A 12/4885MEN1 1049/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.