SCHEMBL6919160

SCHEMBL6919160

COc1ccc(CN2Cc3ccccc3CC2CNC(=O)C(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.51
MTNR1A P48039 4/20 0.44
MTNR1B P49286 4/20 0.44
NQO2 P16083 3/20 0.44
TNF P01375 1/20 0.41
NOD2 Q9HC29 1/20 0.41
NOD1 Q9Y239 1/20 0.41
MMP1 P03956 4/20 0.41
MMP9 P14780 4/20 0.41
MMP3 P08254 3/20 0.41
AREG P15514 2/20 0.41
ADAM17 P78536 2/20 0.41
HDAC8 Q9BY41 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
NR1D1 P20393 1/20 0.40
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7127952 0.77 SIGMAR1 (0.47) OPRM1
SCHEMBL6920302 0.74 HDAC8 (0.53) OPRM1MMP1MMP9MMP3ADAM17
SCHEMBL6920539 0.74 HTR1A (0.50) OPRM1TNFNOD2NOD1MMP1
SCHEMBL6919911 0.73 OPRM1 (0.47) OPRM1OPRD1OPRK1NR1D1
SCHEMBL6820388 0.71 HDAC8 (0.48) MMP1MMP9MMP3AREGADAM17
SCHEMBL17231980 0.69 PPARD (0.47) TNFNOD2NOD1HDAC8DRD2
SCHEMBL29538605 0.68 HDAC8 (0.49) HDAC8OPRK1DRD4
SCHEMBL506516 0.68 HDAC3 (0.60)
SCHEMBL4825496 0.68 SIGMAR1 (0.50) OPRM1OPRD1OPRK1
SCHEMBL32676928 0.67 NAMPT (0.47) OPRM1MMP3OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004041816-A1 AZACYCLIC COMPOUNDS AS OREXIN RECEPTOR ANTAGONIST GLAXO GROUP LIMITED (GB) 2004-05-21 WO disclosed