SCHEMBL6935009

SCHEMBL6935009

CC1(C)CC(NS(C)(=O)=O)c2cc([N+](=O)[O-])ccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.39
CHRNB4 P30926 3/20 0.39
CHRNA3 P32297 3/20 0.39
ALDH1A1 P00352 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
MAPT P10636 2/20 0.39
TSHR P16473 2/20 0.39
PTGS1 P23219 2/20 0.39
PTGS2 P35354 2/20 0.39
PTGES O14684 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALOX15 P16050 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSP90AA1 P07900 1/20 0.38
HIF1A Q16665 2/20 0.38
CHRNA4 P43681 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8182657 0.75 MEN1 (0.46) CYP19A1CHRNB4CHRNA3ALDH1A1MEN1
SCHEMBL6931992 0.75 CYP19A1 (0.40) CYP19A1CHRNB4CHRNA3ALDH1A1CYP1A2
SCHEMBL9156355 0.75 HIF1A (0.46) CHRNB4CHRNA3ALDH1A1MEN1KMT2A
SCHEMBL6938882 0.75 CYP3A4 (0.44) CHRNB4CHRNA3ALDH1A1MEN1KMT2A
SCHEMBL27342629 0.72 ALDH1A1 (0.41) CHRNB4CHRNA3ALDH1A1MEN1KMT2A
SCHEMBL6347611 0.70 CYP19A1 (0.41) CYP19A1CHRNB4CHRNA3ALDH1A1MEN1
SCHEMBL6936648 0.69 CYP19A1 (0.40) CYP19A1ALDH1A1SMN1; SMN2MAPTLMNA
SCHEMBL2062385 0.67 INSR (0.41) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL6560790 0.67 SIRT2 (0.44) CHRNB4CHRNA3ALDH1A1MEN1KMT2A
SCHEMBL20704108 0.67 PNMT (0.47) CHRNB4CHRNA3ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915087-B1 Sulfonamide substituted fused five-membered ring compounds, their use as medicaments as well as pharmaceutical compositions containing them AVENTIS PHARMA GMBH (DE) 2003-04-02 EP disclosed
US-6015822-A ANTIULCER, ANTIDIARRHEA, AND ANTIARRHYTHMIA AGENTS; CARDIOVASCULAR AND GASTROINTESTINAL DISORDERS HOECHST MARION ROUSSEL DEUTSCHLAND GMBH (DE) 2000-01-18 US disclosed
EP-0915087-A2 Sulfonamide substituted fused five-membered ring compounds, their use as medicaments as well as pharmaceutical compositions containing them Hoechst Marion Roussel Deutschland GmbH (DE) 1999-05-12 EP disclosed