SCHEMBL6935372

SCHEMBL6935372

N=C(N)Nc1ccc(C(=O)NC(=O)NN[C@@H](CC(=O)O)C(N)=O)cn1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HCAR3 P49019 1/20 0.36
DEGS1 O15121 1/20 0.36
EPHX2 P34913 1/20 0.36
CXCR2 P25025 1/20 0.35
HDAC1 Q13547 1/20 0.34
ITGB3 P05106 4/20 0.34
ITGAV P06756 3/20 0.34
ITGA2B P08514 1/20 0.34
F10 P00742 1/20 0.34
GCK P35557 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6934969 0.77 ITGB3 (0.51) NPC1RAB9AITGB3ITGAVITGA2B
SCHEMBL6941874 0.75 PYGL (0.42) NPC1RAB9AF10
SCHEMBL6941352 0.73 ITGB3 (0.47) ITGB3ITGAVITGA2BF10
SCHEMBL7879691 0.72 ITGB3 (0.56) NPC1RAB9AITGB3ITGAVITGA2B
SCHEMBL6938993 0.68 ITGB3 (0.51) NPC1RAB9AITGB3ITGAVITGA2B
SCHEMBL6937428 0.66 ITGB3 (0.40) ITGB3ITGA2B
SCHEMBL25212859 0.63 HCAR3 (0.53) RAB9AHCAR3DEGS1CXCR2
SCHEMBL7882801 0.63 ALDH1A1 (0.41) HDAC1ITGB3ITGAV
SCHEMBL6937672 0.63 EPHX2 (0.37) EPHX2ITGB3ITGA2B
SCHEMBL7099306 0.62 ITGB3 (0.51) NPC1RAB9AITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1097127-B1 DIACYLHYDRAZINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2003-03-12 EP disclosed
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US disclosed